SCHEMBL28974416

SCHEMBL28974416

CC(C)N1CCN(c2ccc(C[C@H](NC(=O)OC(C)(C)C)C(=O)Nc3ccc(C(=O)O)cc3)cc2)C(=O)C1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.46
CMA1 P23946 1/20 0.43
AKT1 P31749 1/20 0.42
NTRK1 P04629 1/20 0.41
CTSS P25774 7/20 0.41
CTSK P43235 6/20 0.41
CTSB P07858 2/20 0.40
CTSL P07711 1/20 0.40
SCN9A Q15858 4/20 0.40
ITGB3 P05106 1/20 0.40
ITGB1 P05556 1/20 0.40
ITGAV P06756 1/20 0.40
ITGA2B P08514 1/20 0.40
ITGB5 P18084 1/20 0.40
CCKAR P32238 1/20 0.38
CCKBR P32239 1/20 0.38
PABPC1 P11940 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28974421 1.00 HDAC8 (0.46) HDAC8CMA1AKT1NTRK1CTSS
SCHEMBL23466446 0.93 HDAC8 (0.44) HDAC8CMA1AKT1NTRK1CTSS
SCHEMBL23466444 0.93 HDAC8 (0.44) HDAC8CMA1AKT1NTRK1CTSS
SCHEMBL29139664 0.91 HDAC8 (0.44) HDAC8CMA1AKT1NTRK1CTSS
SCHEMBL28974603 0.90 L3MBTL1 (0.49) HDAC8CMA1AKT1NTRK1CTSS
SCHEMBL28974608 0.90 L3MBTL1 (0.49) HDAC8CMA1AKT1NTRK1CTSS
SCHEMBL28974568 0.89 HDAC8 (0.46) HDAC8CMA1AKT1NTRK1CTSS
SCHEMBL28974559 0.89 HDAC8 (0.46) HDAC8CMA1AKT1NTRK1CTSS
SCHEMBL28974567 0.86 HDAC8 (0.44) HDAC8CMA1AKT1NTRK1CTSS
SCHEMBL28974565 0.86 HDAC8 (0.44) HDAC8CMA1AKT1NTRK1CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114728917-B Oxamide derivative, preparation method and medical application thereof 深圳信立泰药业股份有限公司 2023-12-08 CN disclosed
CN-114728917-A Oxamide derivative, preparation method and medical application thereof 深圳信立泰药业股份有限公司 2022-07-08 CN disclosed