SCHEMBL28980969

SCHEMBL28980969

CC(=O)Nc1c(Cl)cc(Nc2nc(Nc3ccc(N4CCN(C)CC4)cc3)ncc2F)cc1Cl

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 10/20 0.64
MAP3K7 O43318 3/20 0.59
EGFR P00533 1/20 0.59
ALK Q9UM73 2/20 0.58
FLT3 P36888 1/20 0.58
BTK Q06187 1/20 0.58
SYK P43405 1/20 0.56
CCNT1 O60563 1/20 0.56
CCNK O75909 1/20 0.56
CYP3A4 P08684 1/20 0.56
CCND3 P30281 1/20 0.56
CDK9 P50750 1/20 0.56
CDK6 Q00534 1/20 0.56
CTSC P53634 1/20 0.54
FGFR1 P11362 1/20 0.54
SRC P12931 1/20 0.54
MAPK1 P28482 1/20 0.54
MAP2K1 Q02750 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31684801 1.00 BRD4 (0.64) BRD4MAP3K7EGFRALKFLT3
SCHEMBL31684751 0.93 ALK (0.68) BRD4MAP3K7EGFRALKFLT3
SCHEMBL28980963 0.93 ALK (0.68) BRD4MAP3K7EGFRALKFLT3
SCHEMBL31684797 0.91 BRD4 (0.66) BRD4MAP3K7EGFRALKFLT3
SCHEMBL28981000 0.91 BRD4 (0.66) BRD4MAP3K7EGFRALKFLT3
SCHEMBL28980979 0.83 MAP3K7 (0.70) BRD4MAP3K7EGFRALKFLT3
SCHEMBL31260251 0.83 MAP3K7 (0.70) BRD4MAP3K7EGFRALKFLT3
SCHEMBL31684799 0.83 MAP3K7 (0.72) BRD4MAP3K7EGFRALKFLT3
SCHEMBL28980964 0.83 MAP3K7 (0.72) BRD4MAP3K7EGFRALKFLT3
SCHEMBL31684793 0.83 MAP3K7 (0.75) BRD4MAP3K7EGFRALKFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115894381-A 2,4,5-trisubstituted pyrimidine compound and preparation method and application thereof 温州医科大学 2023-04-04 CN claimed
CN-115894381-A 2,4,5-trisubstituted pyrimidine compound and preparation method and application thereof 温州医科大学 2023-04-04 CN disclosed