SCHEMBL28980972

SCHEMBL28980972

C/C=C/C(=O)Nc1ccc(Nc2nc(Nc3ccc(N4CCN(C)CC4)cc3)ncc2Cl)cc1Cl

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K7 O43318 4/20 0.67
FGFR1 P11362 2/20 0.67
MAP2K1 Q02750 2/20 0.67
SRC P12931 1/20 0.67
MAPK1 P28482 1/20 0.67
ALK Q9UM73 3/20 0.62
BRD4 O60885 10/20 0.61
SLC2A1 P11166 1/20 0.59
EGFR P00533 2/20 0.59
CHEK1 O14757 1/20 0.59
AURKA O14965 1/20 0.59
DAPK3 O43293 1/20 0.59
JAK2 O60674 1/20 0.59
PRKD3 O94806 1/20 0.59
MAP4K4 O95819 1/20 0.59
PAK4 O96013 1/20 0.59
ABL1 P00519 1/20 0.59
NTRK1 P04629 1/20 0.59
LCK P06239 1/20 0.59
FYN P06241 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31684798 1.00 MAP3K7 (0.67) MAP3K7FGFR1MAP2K1SRCMAPK1
SCHEMBL31684777 0.91 MAP3K7 (0.80) MAP3K7FGFR1MAP2K1SRCMAPK1
SCHEMBL28980982 0.91 MAP3K7 (0.80) MAP3K7FGFR1MAP2K1SRCMAPK1
SCHEMBL28980981 0.90 MAP3K7 (0.66) MAP3K7FGFR1MAP2K1SRCMAPK1
SCHEMBL31684782 0.90 MAP3K7 (0.66) MAP3K7FGFR1MAP2K1SRCMAPK1
SCHEMBL28980991 0.90 MAP3K7 (0.70) MAP3K7FGFR1MAP2K1SRCMAPK1
SCHEMBL31684780 0.90 MAP3K7 (0.70) MAP3K7FGFR1MAP2K1SRCMAPK1
SCHEMBL31684799 0.88 MAP3K7 (0.72) MAP3K7FGFR1MAP2K1SRCMAPK1
SCHEMBL28980964 0.88 MAP3K7 (0.72) MAP3K7FGFR1MAP2K1SRCMAPK1
SCHEMBL31684761 0.88 MAP3K7 (0.65) MAP3K7FGFR1MAP2K1SRCMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115894381-A 2,4,5-trisubstituted pyrimidine compound and preparation method and application thereof 温州医科大学 2023-04-04 CN claimed
CN-115894381-A 2,4,5-trisubstituted pyrimidine compound and preparation method and application thereof 温州医科大学 2023-04-04 CN disclosed