SCHEMBL28980987

SCHEMBL28980987

CN1CCN(c2ccc(Nc3ncc(F)c(Nc4ccc(NC(=O)c5ccccc5)c(Cl)c4)n3)cc2)CC1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 6/20 0.77
AURKA O14965 4/20 0.65
AURKB Q96GD4 3/20 0.65
FLT3 P36888 1/20 0.62
BTK Q06187 1/20 0.62
ALK Q9UM73 1/20 0.61
CDK2 P24941 2/20 0.59
JAK1 P23458 1/20 0.58
MAP3K7 O43318 3/20 0.57
EGFR P00533 2/20 0.57
FGFR1 P11362 1/20 0.57
SRC P12931 1/20 0.57
MAPK1 P28482 1/20 0.57
MAP2K1 Q02750 1/20 0.57
CCNT1 O60563 1/20 0.56
CCNE1 P24864 1/20 0.56
CDK9 P50750 1/20 0.56
SYK P43405 1/20 0.56
LCK P06239 1/20 0.55
KDR P35968 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31684795 1.00 BRD4 (0.77) BRD4AURKAAURKBFLT3BTK
SCHEMBL28981000 0.89 BRD4 (0.66) BRD4FLT3BTKALKMAP3K7
SCHEMBL31684797 0.89 BRD4 (0.66) BRD4FLT3BTKALKMAP3K7
SCHEMBL17526046 0.87 BRD4 (1.00) BRD4AURKAAURKBFLT3BTK
SCHEMBL28980979 0.87 MAP3K7 (0.70) BRD4AURKAAURKBFLT3BTK
SCHEMBL31260251 0.87 MAP3K7 (0.70) BRD4AURKAAURKBFLT3BTK
SCHEMBL28980969 0.82 BRD4 (0.64) BRD4FLT3BTKALKMAP3K7
SCHEMBL28876170 0.82 BRD4 (0.72) BRD4FLT3BTKCDK2EGFR
SCHEMBL31684801 0.82 BRD4 (0.64) BRD4FLT3BTKALKMAP3K7
SCHEMBL29463626 0.82 BRD4 (0.72) BRD4FLT3BTKCDK2EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115894381-A 2,4,5-trisubstituted pyrimidine compound and preparation method and application thereof 温州医科大学 2023-04-04 CN claimed
CN-115894381-A 2,4,5-trisubstituted pyrimidine compound and preparation method and application thereof 温州医科大学 2023-04-04 CN disclosed