SCHEMBL289838

SCHEMBL289838

CCOC(=O)c1sc(-c2ccc(-c3cccc(C(C)=O)c3)s2)nc1C

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.57
KDM4E B2RXH2 3/20 0.57
CDC7 O00311 4/20 0.53
DBF4 Q9UBU7 4/20 0.53
LMNA P02545 1/20 0.53
MAPT P10636 5/20 0.47
TRPM8 Q7Z2W7 3/20 0.47
KMT2A Q03164 3/20 0.47
MEN1 O00255 2/20 0.47
KIFC1 Q9BW19 4/20 0.47
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
CYP1A2 P05177 1/20 0.47
GAA P10253 1/20 0.47
CYP2C19 P33261 1/20 0.47
HPGD P15428 2/20 0.45
HSD17B10 Q99714 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3619382 0.90 CDC7 (0.62) ALDH1A1KDM4ECDC7DBF4LMNA
SCHEMBL290210 0.88 KDM4E (0.60) ALDH1A1KDM4ECDC7DBF4LMNA
SCHEMBL289156 0.87 ALDH1A1 (0.65) ALDH1A1KDM4ECDC7DBF4LMNA
SCHEMBL290101 0.86 ALDH1A1 (0.64) ALDH1A1KDM4ECDC7DBF4LMNA
SCHEMBL289325 0.86 TRPM8 (0.65) ALDH1A1KDM4ECDC7DBF4LMNA
SCHEMBL290050 0.86 ALDH1A1 (0.58) ALDH1A1KDM4ECDC7DBF4LMNA
SCHEMBL289979 0.86 TRPM8 (0.65) ALDH1A1KDM4ECDC7DBF4LMNA
SCHEMBL289696 0.84 ALDH1A1 (0.56) ALDH1A1KDM4ECDC7DBF4LMNA
SCHEMBL290128 0.84 MAPT (0.69) ALDH1A1KDM4ECDC7DBF4LMNA
SCHEMBL290226 0.83 KDM4E (0.55) ALDH1A1KDM4ECDC7DBF4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427447-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION Pike Pharma GmbH (CH) 2012-03-14 EP disclosed
WO-2010128163-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION PIKE PHARMA GMBH (CH) 2010-11-11 WO disclosed