SCHEMBL28984072

SCHEMBL28984072

Cn1nc(N2CCC(=O)NC2=O)c2cccc(N)c21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 17/20 1.00
DDB1 Q16531 16/20 1.00
MEN1 O00255 1/20 0.34
USP2 O75604 1/20 0.34
KMT2A Q03164 1/20 0.34
ATM Q13315 1/20 0.34
KEAP1 Q14145 1/20 0.34
NFE2L2 Q16236 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30472890 1.00 CRBN (1.00) CRBNDDB1MEN1USP2KMT2A
SCHEMBL25578237 0.89 CRBN (0.80) CRBNDDB1
SCHEMBL25026932 0.87 CRBN (0.77) CRBNDDB1
SCHEMBL25595586 0.86 CRBN (0.76) CRBNDDB1
SCHEMBL25567340 0.84 CRBN (0.72) CRBNDDB1
SCHEMBL25566821 0.84 CRBN (0.72) CRBNDDB1
SCHEMBL30472913 0.84 CRBN (0.72) CRBNDDB1MEN1USP2KMT2A
SCHEMBL26826457 0.83 CRBN (1.00) CRBNDDB1
SCHEMBL30258522 0.83 CRBN (1.00) CRBNDDB1
SCHEMBL31443986 0.82 CRBN (0.69) CRBNDDB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115968293-A Cereblon binding compounds, compositions thereof, and methods of use thereof for treatment 新基公司 2023-04-14 CN disclosed