SCHEMBL25567340

SCHEMBL25567340

CC(C)c1cccc2c(N3CCC(=O)NC3=O)nn(C)c12

nearest known ligand 0.72

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 19/20 0.72
DDB1 Q16531 18/20 0.72
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27323325 0.90 CRBN (0.58) CRBNDDB1KDM4EALDH1A1HPGD
SCHEMBL28984072 0.84 CRBN (1.00) CRBNDDB1
SCHEMBL25026932 0.84 CRBN (0.77) CRBNDDB1
SCHEMBL30472890 0.84 CRBN (1.00) CRBNDDB1
SCHEMBL25595606 0.84 CRBN (0.60) CRBNDDB1KDM4EALDH1A1HPGD
SCHEMBL25595586 0.83 CRBN (0.76) CRBNDDB1
SCHEMBL25578237 0.83 CRBN (0.80) CRBNDDB1
SCHEMBL25567342 0.81 CRBN (0.54) CRBNDDB1KDM4EALDH1A1HPGD
SCHEMBL30472913 0.81 CRBN (0.72) CRBNDDB1
SCHEMBL25566821 0.81 CRBN (0.72) CRBNDDB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023244918-A1 QUINOLONE BCL6 BIFUNCTIONAL DEGRADERS Treeline Biosciences, Inc. (US) 2023-12-21 WO disclosed
WO-2023240038-A1 TRICYCLIC QUINOLONE BCL6 BIFUNCTIONAL DEGRADERS Treeline Biosciences, Inc. (US) 2023-12-14 WO disclosed
WO-2023083194-A1 WEE1 PROTEIN KINASE DEGRADATION AGENT AND USE THEREOF 杭州格博生物医药有限公司 2023-05-19 WO disclosed