SCHEMBL28985195

SCHEMBL28985195

CC(/C=C/c1ccccc1)c1ccc(-c2ccc(C(F)(F)F)cc2)cn1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.42
CYP1A1 P04798 1/20 0.38
MAOB P27338 1/20 0.38
CYP1B1 Q16678 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
SCN2A Q99250 2/20 0.37
CYP19A1 P11511 1/20 0.37
TRPV1 Q8NER1 3/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
PDE2A O00408 1/20 0.34
CDC25B P30305 1/20 0.33
DUSP3 P51452 1/20 0.33
PTGES2 Q9H7Z7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28985164 0.88 GRM5 (0.36) CA1NPC1RAB9A
SCHEMBL28985166 0.88 GRM5 (0.36) CA1NPC1RAB9A
SCHEMBL30475177 0.88 GRM5 (0.36) CA1NPC1RAB9A
SCHEMBL28985198 0.82 ALDH1A1 (0.38) GRIN1GRIN2B
SCHEMBL28985196 0.82 ALDH1A1 (0.38) GRIN1GRIN2B
SCHEMBL30475181 0.76 GRM5 (0.45) NPC1
SCHEMBL2609357 0.76 KIF11 (0.47) KIF11SCN2A
SCHEMBL30475167 0.75 S1PR2 (0.38) CYP1B1NPC1RAB9A
SCHEMBL28985165 0.75 S1PR2 (0.38) CYP1B1NPC1RAB9A
SCHEMBL28985169 0.75 S1PR2 (0.38) CYP1B1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115974927-A Diamine-derived phosphine chiral phosphine oxide ligand-promoted nickel-catalyzed asymmetric alkylation of pyridine C2-H bond 南开大学 2023-04-18 CN disclosed