SCHEMBL28986232

SCHEMBL28986232

Nc1ncc2[nH]cc(-c3cc(I)ccc3F)c2n1

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAP3K14 Q99558 10/20 0.50
MAPKAPK2 P49137 2/20 0.49
CLK1 P49759 7/20 0.41
CDK5 Q00535 4/20 0.41
CDK5R1 Q15078 4/20 0.41
TDO2 P48775 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30219604 1.00 MAP3K14 (0.50) MAP3K14MAPKAPK2CLK1CDK5CDK5R1
SCHEMBL1612797 0.76 DHFR (0.45)
SCHEMBL25247947 0.68 MAP3K14 (1.00) MAP3K14
SCHEMBL25247949 0.68 MAP3K14 (1.00) MAP3K14
SCHEMBL28986332 0.67 MAPKAPK2 (0.60) MAP3K14MAPKAPK2CLK1CDK5CDK5R1
SCHEMBL30219627 0.67 MAPKAPK2 (0.60) MAP3K14MAPKAPK2CLK1CDK5CDK5R1
SCHEMBL30219575 0.66 MAP3K14 (0.54) MAP3K14MAPKAPK2CLK1CDK5CDK5R1
SCHEMBL28986214 0.66 MAP3K14 (0.54) MAP3K14MAPKAPK2CLK1CDK5CDK5R1
SCHEMBL19671051 0.64 MAPKAPK2 (0.46) MAP3K14MAPKAPK2CLK1CDK5CDK5R1
SCHEMBL15730201 0.64 MAPKAPK2 (0.46) MAP3K14MAPKAPK2CLK1CDK5CDK5R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109810110-B Compound with 2-aminopyrimidine structure, preparation method and application thereof 中国科学院上海药物研究所 2023-01-24 CN disclosed