SCHEMBL28987478

SCHEMBL28987478

CN1C(=O)CNCC1C(=O)OC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.35
CASP3 P42574 1/20 0.33
BRD4 O60885 1/20 0.32
CHRM2 P08172 1/20 0.31
CHRM1 P11229 1/20 0.31
CHRM3 P20309 1/20 0.31
PLA2G10 O15496 1/20 0.31
PLA2G5 P39877 1/20 0.31
GAA P10253 1/20 0.31
KDM4E B2RXH2 1/20 0.30
MAPT P10636 1/20 0.30
THRB P10828 1/20 0.30
NFKB1 P19838 1/20 0.30
NFKB2 Q00653 1/20 0.30
RELA Q04206 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25334933 0.82 BRD4 (0.41) BRD4
Hydrochloric Acid SCHEMBL30515108 0.81 BRD4 (0.40) BRD4
SCHEMBL1637463 0.79 P2RX7 (0.40) MAPK1CASP3PLA2G10PLA2G5GAA
SCHEMBL14814407 0.79 P2RX7 (0.40) MAPK1CASP3PLA2G10PLA2G5GAA
SCHEMBL24750243 0.76 P2RX7 (0.40) MAPK1CHRM2CHRM1CHRM3
SCHEMBL23230738 0.76 P2RX7 (0.40) MAPK1CHRM2CHRM1CHRM3
SCHEMBL29060344 0.74 MAPK1 (0.30) MAPK1
SCHEMBL7393196 0.71 HRH3 (0.33) MAPK1CASP3
SCHEMBL6634675 0.70 MAPK1 (0.38) MAPK1GAAKDM4EMAPTTHRB
SCHEMBL1637995 0.69 P2RX7 (0.40) MAPK1BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115996927-A Pyrimido [5,4-d ] pyrimidine derivatives and combinations with adenosine receptor antagonists as ENT inhibitors for the treatment of cancer ITEOS比利时公司 2023-04-21 CN disclosed