SCHEMBL28989394

SCHEMBL28989394

CCCC(N=C(c1ccccc1)c1ccccc1)C(=O)Oc1ccc(Cl)nn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 1/20 0.44
LMNA P02545 3/20 0.34
KMT2A Q03164 3/20 0.34
POLB P06746 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A3 Q01959 1/20 0.33
MEN1 O00255 2/20 0.32
PGR P06401 1/20 0.32
ADRA2A P08913 1/20 0.32
ADRA2B P18089 1/20 0.32
HTR2A P28223 1/20 0.32
HRH1 P35367 1/20 0.32
KCNH2 Q12809 1/20 0.32
CES2 O00748 1/20 0.31
CES1 P23141 1/20 0.31
PRSS1 P07477 1/20 0.31
CTSG P08311 1/20 0.31
CTRB1 P17538 1/20 0.31
CMA1 P23946 1/20 0.31
PPARG P37231 4/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14493754 0.76 AAK1 (0.54) AAK1LMNAKMT2APOLBSLC6A2
SCHEMBL28614576 0.76 AAK1 (0.45) AAK1LMNANPC1ALDH1A1SMN1; SMN2
SCHEMBL24982012 0.74 AAK1 (0.40) AAK1KMT2AMEN1NPC1ALDH1A1
SCHEMBL26693677 0.73 KMT2A (0.41) AAK1LMNAKMT2AMEN1NPC1
SCHEMBL16116863 0.73 AAK1 (0.76) AAK1LMNAKMT2APOLBSLC6A2
SCHEMBL20786122 0.70 AAK1 (0.47) AAK1LMNAKMT2APOLBSLC6A2
SCHEMBL29154278 0.70 LMNA (0.40) AAK1LMNAKMT2APOLBALDH1A1
SCHEMBL9667964 0.69 AAK1 (0.53) AAK1LMNAPRSS1CTSGCTRB1
SCHEMBL24982015 0.68 ALDH1A1 (0.40) AAK1KMT2APOLBMEN1ALDH1A1
SCHEMBL8199100 0.67 AAK1 (0.50) AAK1LMNAKMT2APOLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115996923-A Nitrile derivative as dipeptidyl peptidase 1 inhibitor and application thereof 四川海思科制药有限公司 2023-04-21 CN disclosed