SCHEMBL28989707

SCHEMBL28989707

NCCCOc1ccc2c(c1)c(-c1c[c]ccc1)nn2C1CCCCO1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DNMT3A Q9Y6K1 1/20 0.35
AVPR1B P47901 2/20 0.35
CYP4F2 P78329 4/20 0.33
CYP4A11 Q02928 4/20 0.33
SIGMAR1 Q99720 1/20 0.33
PSMB5 P28074 2/20 0.31
PSMB1 P20618 1/20 0.31
RXRA P19793 1/20 0.31
RXRB P28702 1/20 0.31
RXRG P48443 1/20 0.31
HTR1A P08908 1/20 0.30
HTR1D P28221 1/20 0.30
HTR1B P28222 1/20 0.30
ATR Q13535 1/20 0.30
PLA2G2A P14555 2/20 0.30
RET P07949 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30242664 0.84 DNMT3A (0.38) DNMT3AAVPR1BCYP4F2CYP4A11SIGMAR1
SCHEMBL24012720 0.84 DNMT3A (0.38) DNMT3AAVPR1BCYP4F2CYP4A11SIGMAR1
SCHEMBL30242637 0.80 CMKLR1 (0.35) DNMT3AAVPR1BCYP4F2CYP4A11SIGMAR1
SCHEMBL24012969 0.80 CMKLR1 (0.35) DNMT3AAVPR1BCYP4F2CYP4A11SIGMAR1
SCHEMBL30242538 0.80 CYP4F2 (0.35) DNMT3AAVPR1BCYP4F2CYP4A11RXRA
SCHEMBL24012616 0.80 CYP4F2 (0.35) DNMT3AAVPR1BCYP4F2CYP4A11RXRA
SCHEMBL24012651 0.80 LSS (0.38) AVPR1BCYP4F2CYP4A11HTR1AHTR1D
SCHEMBL24012649 0.80 CYP4F2 (0.40) AVPR1BCYP4F2CYP4A11SIGMAR1RXRA
SCHEMBL5648303 0.78 RXRA (0.32) DNMT3ARXRARXRBRXRGATR
SCHEMBL24013099 0.78 CMKLR1 (0.37) CYP4F2CYP4A11RETHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115996932-A New macrocyclic LRRK2 kinase inhibitors 法国施维雅药厂 2023-04-21 CN disclosed