SCHEMBL289901

SCHEMBL289901

COCCn1c(=O)sc2ccc(-c3ccc(CC(C#N)C4CC(C(N)=O)CCO4)cc3)cc21

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSC P53634 16/20 0.55
KCNH2 Q12809 1/20 0.42
PPARA Q07869 1/20 0.33
DPP4 P27487 1/20 0.32
PPARG P37231 1/20 0.32
CTSK P43235 2/20 0.32
GAA P10253 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL288983 0.86 CTSC (0.55) CTSCKCNH2
SCHEMBL290060 0.81 CTSC (0.58) CTSCKCNH2
SCHEMBL289754 0.79 CTSC (0.52) CTSCKCNH2CTSK
SCHEMBL289902 0.79 CTSC (0.72) CTSCKCNH2CTSK
SCHEMBL290338 0.78 CTSC (0.44) CTSCDPP4
SCHEMBL299868 0.76 CTSC (0.47) CTSCCTSK
SCHEMBL289369 0.76 CTSC (0.53) CTSCCTSK
SCHEMBL288811 0.75 CTSC (0.49) CTSCDPP4
SCHEMBL290171 0.75 CTSC (0.45) CTSCCTSK
SCHEMBL289986 0.75 CTSC (0.42) CTSCDPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427445-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 AstraZeneca AB (SE) 2012-03-14 EP claimed
EP-2427445-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 AstraZeneca AB (SE) 2012-03-14 EP disclosed