SCHEMBL28991129

SCHEMBL28991129

CCOC(=O)c1nn(Cc2ccc(F)cc2)c(Cl)c1C=COC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.44
NPC1 O15118 2/20 0.42
LMNA P02545 2/20 0.42
RAB9A P51151 1/20 0.42
PDE4A P27815 2/20 0.41
PDE4B Q07343 2/20 0.41
PDE4C Q08493 2/20 0.41
PDE4D Q08499 2/20 0.41
ALDH1A1 P00352 3/20 0.41
ELANE P08246 1/20 0.40
CYP19A1 P11511 2/20 0.39
MAPT P10636 4/20 0.39
TP53 P04637 1/20 0.39
HPGD P15428 1/20 0.39
MEN1 O00255 1/20 0.39
STAT3 P40763 1/20 0.39
STAT1 P42224 1/20 0.39
KMT2A Q03164 1/20 0.39
POLB P06746 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30076384 1.00 KDM4E (0.44) KDM4ENPC1LMNARAB9APDE4A
SCHEMBL23081412 0.91 P2RX7 (0.39) KDM4ENPC1LMNARAB9APDE4A
SCHEMBL25974658 0.91 P2RX7 (0.39) KDM4ENPC1LMNARAB9APDE4A
SCHEMBL20477230 0.89 CYP19A1 (0.50) KDM4ELMNARAB9APDE4APDE4B
SCHEMBL20477228 0.89 CYP19A1 (0.50) KDM4ELMNARAB9APDE4APDE4B
SCHEMBL23081613 0.87 P2RX7 (0.35) KDM4ENPC1LMNARAB9APDE4A
SCHEMBL30121872 0.87 ALDH1A1 (0.41) NPC1LMNARAB9AALDH1A1ELANE
SCHEMBL23070389 0.87 TSHR (0.39) KDM4ENPC1LMNARAB9AELANE
SCHEMBL23070390 0.87 TSHR (0.39) KDM4ENPC1LMNARAB9AELANE
SCHEMBL28991056 0.87 KDM4E (0.47) KDM4ENPC1LMNARAB9APDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115867557-B Azepine condensed ring compound and medical application thereof 中国医药研究开发中心有限公司 2025-02-18 CN disclosed
CN-115867557-A Azepine fused ring compounds and medical application thereof 中国医药研究开发中心有限公司 2023-03-28 CN disclosed
WO-2022237890-A1 AZEPINE-TYPE FUSED RING COMPOUND AND PHARMACEUTICAL USE THEREOF 中国医药研究开发中心有限公司 2022-11-17 WO disclosed