SCHEMBL28995145

SCHEMBL28995145

CC(C)(C)C(=O)On1ccc2c(-c3cn[nH]c3)ncnc21

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.38
JAK2 O60674 4/20 0.37
P2RX7 Q99572 1/20 0.33
NAMPT P43490 1/20 0.33
PIK3CD O00329 1/20 0.33
CYP3A4 P08684 1/20 0.32
PRMT5 O14744 1/20 0.32
KDM5B Q9UGL1 1/20 0.31
JAK3 P52333 1/20 0.31
ROCK2 O75116 2/20 0.31
CHUK O15111 1/20 0.31
NTRK1 P04629 1/20 0.31
CSNK1D P48730 1/20 0.31
CSNK1E P49674 1/20 0.31
RET P07949 1/20 0.30
PDPK1 O15530 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17967357 0.89 SIGMAR1 (0.38) SIGMAR1JAK2P2RX7NAMPTPIK3CD
SCHEMBL871452 0.81 SIGMAR1 (0.39) SIGMAR1JAK2P2RX7NAMPTPIK3CD
SCHEMBL30749810 0.81 SIGMAR1 (0.39) SIGMAR1JAK2P2RX7NAMPTPIK3CD
SCHEMBL31291536 0.79 SIGMAR1 (0.37) SIGMAR1JAK2P2RX7NAMPTCYP3A4
SCHEMBL30945101 0.76 SIGMAR1 (0.38) SIGMAR1JAK2NAMPTPRMT5ROCK2
SCHEMBL28861111 0.75 SLC22A12 (0.43) JAK2P2RX7PRMT5
SCHEMBL13058244 0.75 SIGMAR1 (0.48) SIGMAR1JAK2PIK3CDCYP3A4PRMT5
SCHEMBL24205668 0.75 SIGMAR1 (0.44) SIGMAR1JAK2P2RX7PRMT5JAK3
SCHEMBL13286026 0.73 SIGMAR1 (0.38) SIGMAR1JAK2P2RX7PIK3CD
SCHEMBL10222870 0.72 SIGMAR1 (0.45) SIGMAR1P2RX7PRMT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115856141-A Method for separating and determining tinib key intermediate and related impurities thereof by HPLC 上海博悦生物科技有限公司 2023-03-28 CN disclosed