SCHEMBL28998729

SCHEMBL28998729

Cn1nnc(-c2ncc(NC(=O)c3ccc(Cl)nc3)cc2F)c1OC(N)=O

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNQ3 O43525 15/20 0.48
KCNQ2 O43526 15/20 0.48
KCNE1 P15382 11/20 0.48
KCNQ1 P51787 11/20 0.48
RAB9A P51151 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
BACE1 P56817 1/20 0.43
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
NPC1 O15118 1/20 0.41
POLB P06746 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
KCNQ5 Q9NR82 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28998741 0.87 RAB9A (0.50) KCNQ3KCNQ2KCNE1KCNQ1RAB9A
SCHEMBL28998201 0.86 KCNQ3 (0.38) KCNQ3KCNQ2KCNE1KCNQ1RAB9A
SCHEMBL28998727 0.83 GAA (0.37) KCNQ3KCNQ2KCNE1KCNQ1SMN1; SMN2
SCHEMBL28998183 0.82 JAK2 (0.34) RAB9ASMN1; SMN2BACE1MEN1KMT2A
SCHEMBL28998221 0.79 KMT2A (0.42) KCNQ3KCNQ2KCNE1KCNQ1RAB9A
SCHEMBL24867499 0.75 KCNQ3 (0.42) KCNQ3KCNQ2KCNE1KCNQ1RAB9A
SCHEMBL28998733 0.74 BACE1 (0.39) BACE1
SCHEMBL28998215 0.74
SCHEMBL28998794 0.74
Hydrochloric Acid SCHEMBL28998795 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115942972-A LPA receptor antagonists and uses thereof 吉利德科学公司 2023-04-07 CN disclosed