SCHEMBL28998740

SCHEMBL28998740

COC(=O)Nc1ccc(-c2nnn(C)c2OC(N)=O)nc1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.37
SMN1; SMN2 Q16637 4/20 0.35
TSHR P16473 1/20 0.34
ALDH1A1 P00352 4/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 3/20 0.32
RAB9A P51151 3/20 0.32
NPC1 O15118 2/20 0.32
PTPN1 P18031 1/20 0.32
KMT2A Q03164 3/20 0.32
HPGD P15428 1/20 0.32
GLA P06280 1/20 0.31
MAPKAPK2 P49137 1/20 0.31
F11 P03951 1/20 0.31
POLB P06746 1/20 0.31
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28998220 0.90 MAPT (0.36) KDM4ESMN1; SMN2ALDH1A1MAPTRAB9A
SCHEMBL28998195 0.89 ALDH1A1 (0.41) KDM4ESMN1; SMN2TSHRALDH1A1MAPT
SCHEMBL28998178 0.89 BCL2 (0.41) MAPKAPK2
SCHEMBL28998174 0.88 NPC1 (0.34) KDM4ESMN1; SMN2ALDH1A1MAPTRAB9A
SCHEMBL28998172 0.87 SMN1; SMN2 (0.42) KDM4ESMN1; SMN2TSHRALDH1A1MAPT
SCHEMBL28998224 0.86 CYP1A2 (0.38) SMN1; SMN2ALDH1A1TP53MAPTRAB9A
SCHEMBL28998796 0.85 PTPN1 (0.51) KDM4ESMN1; SMN2MAPTRAB9ANPC1
SCHEMBL28998180 0.84 MEN1 (0.30) KMT2AMEN1
SCHEMBL28998165 0.84 L3MBTL1 (0.39) KDM4ESMN1; SMN2TSHRTP53MAPT
SCHEMBL28998187 0.83 SMN1; SMN2 (0.41) KDM4ESMN1; SMN2TSHRALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115942972-A LPA receptor antagonists and uses thereof 吉利德科学公司 2023-04-07 CN disclosed