SCHEMBL28999960

SCHEMBL28999960

Cn1ncc2c(=O)[nH]c3cc(Br)ccc3c21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 2/20 0.45
METAP2 P50579 1/20 0.41
AXL P30530 2/20 0.40
CDK4 P11802 3/20 0.39
CCND1 P24385 3/20 0.39
CAMK2A Q9UQM7 3/20 0.39
CAMK2B Q13554 2/20 0.39
CAMK2G Q13555 2/20 0.39
CAMK2D Q13557 2/20 0.39
CCNE2 O96020 2/20 0.38
CCNE1 P24864 2/20 0.38
CDK2 P24941 2/20 0.38
TP53 P04637 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
PDE5A O76074 3/20 0.36
EGFR P00533 1/20 0.35
CDK9 P50750 2/20 0.35
CDK5 Q00535 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30273162 1.00 PTGES (0.45) PTGESMETAP2AXLCDK4CCND1
SCHEMBL24099148 0.83 PARP1 (0.48) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL30380737 0.83 PARP1 (0.48) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL30273149 0.82 PARP1 (0.41) ALDH1A1LMNAHPGD
SCHEMBL29203527 0.82 PARP1 (0.41) ALDH1A1LMNAHPGD
SCHEMBL31552856 0.81 TP53 (0.34) TP53PDE5ACDK9CDK5AURKA
SCHEMBL31552840 0.80 PARP1 (0.43) TP53ALDH1A1HPGD
SCHEMBL31386900 0.80 PARP1 (0.55) DYRK1AALDH1A1HPGD
SCHEMBL30273156 0.80 PARP1 (0.50) CDK2DYRK1AALDH1A1LMNAHPGD
SCHEMBL30273077 0.79 PARP1 (0.50) TP53FGFR1FLT1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116075512-A Heterocyclic compounds and imaging agents for imaging huntingtin CHDI基金会股份有限公司 2023-05-05 CN disclosed