SCHEMBL29001083

SCHEMBL29001083

NC(=O)c1cccc2nc(O)c(O)nc12

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 17/20 0.51
ALDH1A1 P00352 2/20 0.49
PARP2 Q9UGN5 2/20 0.47
KDM4E B2RXH2 1/20 0.44
MAPT P10636 1/20 0.44
HPGD P15428 1/20 0.44
TSHR P16473 1/20 0.44
HSD17B10 Q99714 1/20 0.44
PARP3 Q9Y6F1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30380155 1.00 PARP1 (0.51) PARP1ALDH1A1PARP2KDM4EMAPT
SCHEMBL10868710 0.86 ALDH1A1 (0.58) PARP1ALDH1A1PARP2PARP3
SCHEMBL818929 0.83 ALDH1A1 (0.70) PARP1ALDH1A1PARP2MAPTPARP3
SCHEMBL10555620 0.83 ALDH1A1 (0.70) PARP1ALDH1A1KDM4EMAPTHPGD
SCHEMBL29611021 0.83 ALDH1A1 (0.70) PARP1ALDH1A1PARP2MAPTPARP3
SCHEMBL2624160 0.82 PARP1 (0.51) PARP1ALDH1A1PARP2
SCHEMBL28274572 0.82 ACHE (0.57) PARP1ALDH1A1PARP2KDM4EMAPT
SCHEMBL26523348 0.81 ALDH1A1 (0.49) PARP1ALDH1A1KDM4EMAPT
SCHEMBL2606618 0.80 PARP1 (0.56) PARP1ALDH1A1PARP2
SCHEMBL8411208 0.79 PARP1 (0.54) PARP1ALDH1A1PARP2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116134026-A Triazole derivatives and their use as tankyrase inhibitors 奥斯陆大学国家医院 2023-05-16 CN disclosed