SCHEMBL29005126

SCHEMBL29005126

CCOC(=O)c1ccn(C(F)C(F)F)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.45
KDM4E B2RXH2 3/20 0.41
POLB P06746 1/20 0.41
JMJD6 Q6NYC1 2/20 0.40
MAPK1 P28482 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
KMT2A Q03164 1/20 0.39
TSHR P16473 2/20 0.39
PDE4D Q08499 1/20 0.39
GAA P10253 1/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24915026 0.88 CYP1A2 (0.47) CYP1A2KDM4EPOLBJMJD6MAPK1
SCHEMBL1058997 0.83 CYP1A2 (0.49) CYP1A2KDM4EPOLBJMJD6MAPK1
SCHEMBL29052704 0.78 ALDH1A1 (0.32) NPC1RAB9AALDH1A1SMN1; SMN2MAPT
SCHEMBL22125629 0.77 CYP1A2 (0.43) CYP1A2KDM4EPOLBJMJD6MAPK1
SCHEMBL29224345 0.77 ALDH1A1 (0.49) CYP1A2KDM4EPOLBMAPK1CA12
SCHEMBL6444656 0.77 CYP1A2 (0.45) CYP1A2KDM4EPOLBJMJD6NPC1
SCHEMBL10436784 0.76 KMT2A (0.56) CYP1A2KDM4EPOLBJMJD6MAPK1
SCHEMBL23234117 0.76 CYP1A2 (0.53) CYP1A2KDM4EMAPK1NPC1RAB9A
SCHEMBL10817921 0.76 TSHR (0.60) CYP1A2KDM4EPOLBJMJD6MAPK1
SCHEMBL29005141 0.76 SMN1; SMN2 (0.36) KDM4EPOLBTSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117881661-A Condensed heterocyclic derivative 杨森科学爱尔兰无限公司 2024-04-12 CN disclosed
CN-117715909-A Condensed heterocyclic derivative 杨森科学爱尔兰无限公司 2024-03-15 CN disclosed
CN-116134018-A 2-oxoimidazolidine-4-carboxamide as NAV1.8 inhibitor 默沙东有限责任公司 2023-05-16 CN disclosed