SCHEMBL29007155

SCHEMBL29007155

COc1ccc2c(c1)ncn2-c1nccc(Nc2ccc(-c3cnn(COCC[Si](C)(C)C)c3)cc2)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 1/20 0.45
ROCK2 O75116 3/20 0.41
ROCK1 Q13464 1/20 0.41
ABL1 P00519 12/20 0.38
CSF1R P07333 12/20 0.38
LYN P07948 12/20 0.38
SIK1 P57059 12/20 0.38
SIK2 Q9H0K1 12/20 0.38
SIK3 Q9Y2K2 12/20 0.38
PRKAB2 O43741 11/20 0.38
PRKAG1 P54619 11/20 0.38
PRKAA1 Q13131 11/20 0.38
TGFBR1 P36897 10/20 0.38
TGFBR2 P37173 9/20 0.38
FGFR1 P11362 1/20 0.35
KDR P35968 1/20 0.35
KDM4E B2RXH2 2/20 0.34
NPC1 O15118 2/20 0.34
ALDH1A1 P00352 2/20 0.34
MAPT P10636 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28777048 0.94 LCK (0.45) LCKROCK2ROCK1ABL1CSF1R
SCHEMBL29674607 0.88 ROCK2 (0.42) LCKROCK2ROCK1NPC1ALDH1A1
SCHEMBL28777015 0.88 ROCK2 (0.42) LCKROCK2ROCK1NPC1ALDH1A1
SCHEMBL28777011 0.86 ROCK2 (0.42) LCKROCK2ROCK1KDRNPC1
SCHEMBL16637702 0.85 ROCK2 (0.44) ROCK2ROCK1KDRNPC1ALDH1A1
SCHEMBL16637704 0.82 ROCK2 (0.65) ROCK2ROCK1
SCHEMBL29674711 0.78 MEN1 (0.43) ROCK2ROCK1KDRNPC1ALDH1A1
SCHEMBL29674733 0.78 MEN1 (0.43) ROCK2ROCK1KDRNPC1ALDH1A1
SCHEMBL29674761 0.78 ROCK2 (0.65) LCKROCK2ROCK1
SCHEMBL29007158 0.78 ROCK2 (0.65) LCKROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114573566-B Selective ROCK2 kinase inhibitors 杭州邦顺制药有限公司 2023-05-30 CN disclosed