SCHEMBL29014159

SCHEMBL29014159

Fc1[c]c(-c2nccs2)ccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.44
LOXL2 Q9Y4K0 1/20 0.40
CYP2A6 P11509 1/20 0.40
HSP90AA1 P07900 1/20 0.39
CYP1A1 P04798 3/20 0.37
CYP1A2 P05177 3/20 0.37
CYP1B1 Q16678 3/20 0.37
RAB9A P51151 2/20 0.37
ADORA2A P29274 2/20 0.35
ADORA1 P30542 2/20 0.35
METAP1 P53582 1/20 0.35
KMT2A Q03164 2/20 0.35
NPC1 O15118 1/20 0.35
PKM P14618 1/20 0.35
SYK P43405 2/20 0.34
ADRB2 P07550 1/20 0.33
F2RL1 P55085 1/20 0.33
CASP6 P55212 1/20 0.32
SRC P12931 1/20 0.31
CDK2 P24941 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1671008 0.71 ADRB2 (0.32) CYP2A6ADRB2
SCHEMBL2342778 0.70 PDPK1 (0.47) PDPK1LOXL2CYP2A6HSP90AA1RAB9A
SCHEMBL578376 0.70 PDPK1 (0.52) PDPK1LOXL2CYP2A6HSP90AA1CYP1A2
SCHEMBL28020115 0.69 PDPK1 (0.50) PDPK1LOXL2CYP2A6HSP90AA1CYP1A1
SCHEMBL4721859 0.69 RAB9A (0.49) PDPK1LOXL2CYP2A6HSP90AA1RAB9A
SCHEMBL29118010 0.68 KDM4E (0.41) CYP2A6CYP1A2RAB9AKMT2ANPC1
SCHEMBL29014149 0.67 KDM4E (0.48) CYP2A6HSP90AA1CYP1A2RAB9AMETAP1
SCHEMBL28045453 0.67 PDPK1 (0.39) PDPK1LOXL2CYP2A6HSP90AA1CYP1A1
SCHEMBL4719613 0.66 RAB9A (0.45) PDPK1LOXL2CYP2A6HSP90AA1CYP1A1
SCHEMBL102331 0.66 PDPK1 (0.59) PDPK1LOXL2CYP2A6HSP90AA1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116217593-A Octahydropyrrolo [3,4-c ] pyrrole methyl ketone derivative and application thereof 江苏恩华药业股份有限公司 2023-06-06 CN disclosed