SCHEMBL29014181

SCHEMBL29014181

O=C(O)c1c(F)cccc1-c1nccs1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.51
HCRTR2 O43614 2/20 0.51
KMT2A Q03164 2/20 0.44
PDPK1 O15530 1/20 0.42
CTSA P10619 2/20 0.40
AR P10275 1/20 0.40
MGAM O43451 3/20 0.40
GAA P10253 3/20 0.40
SI P14410 3/20 0.40
MGAM2 Q2M2H8 3/20 0.40
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
VCP P55072 1/20 0.39
CASP6 P55212 1/20 0.38
ECE1 P42892 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29014160 0.80 HCRTR1 (0.48) HCRTR1HCRTR2KMT2ACTSAAR
SCHEMBL30960750 0.79 HCRTR1 (0.45) HCRTR1HCRTR2KMT2ACTSAAR
SCHEMBL8567274 0.78 PDPK1 (0.55) HCRTR1HCRTR2PDPK1ARMGAM
SCHEMBL30960727 0.76 ALB (0.45) KMT2APDPK1CTSAMGAMGAA
SCHEMBL29228640 0.76 CES2 (0.39) KMT2ACES2CES1KDM4EALDH1A1
SCHEMBL29228633 0.76 ALB (0.45) KMT2APDPK1CTSAMGAMGAA
SCHEMBL1586160 0.76 HCRTR1 (0.45) HCRTR1HCRTR2CES2CES1KDM4E
SCHEMBL28839674 0.75 KDM4E (0.41) PDPK1ECE1PTGDR2KDM4EALDH1A1
SCHEMBL19259537 0.74 HCRTR1 (0.41) HCRTR1HCRTR2KMT2ACTSAECE1
SCHEMBL5698661 0.74 CYP1A2 (0.53) PDPK1GAAECE1PTGDR2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116217593-B Octahydropyrrolo [3,4-c ] pyrrole methyl ketone derivative and application thereof 江苏恩华药业股份有限公司 2025-05-09 CN disclosed
CN-118027018-A Tetrahydrocyclopentyl [ c ] pyrrole methyl ketone derivative, preparation method and application thereof 江苏恩华药业股份有限公司 2024-05-14 CN disclosed
CN-116217593-A Octahydropyrrolo [3,4-c ] pyrrole methyl ketone derivative and application thereof 江苏恩华药业股份有限公司 2023-06-06 CN disclosed