SCHEMBL29014633

SCHEMBL29014633

COCOc1cc(F)c(C2CC2)c(Br)c1

nearest known ligand 0.31

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.31
HTR1A P08908 2/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
EGFR P00533 1/20 0.30
KDR P35968 1/20 0.30
TAAR1 Q96RJ0 1/20 0.30
ROR1 Q01973 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23043281 0.82 HTR1A (0.32) MCHR1HTR1AROR1
SCHEMBL29680450 0.82 HTR1A (0.32) MCHR1HTR1AROR1
SCHEMBL30033055 0.73
SCHEMBL29233776 0.72 FFAR1 (0.38)
SCHEMBL23043192 0.72 TAAR1 (0.32) TAAR1
SCHEMBL31108404 0.71 NR3C1 (0.33) ROR1
SCHEMBL26604856 0.70 TAAR1 (0.36) TAAR1
SCHEMBL2171833 0.70 EGFR (0.43) MCHR1KDM4EALDH1A1EGFRKDR
SCHEMBL19616678 0.70 KDM4E (0.36) KDM4EALDH1A1EGFRKDR
SCHEMBL29887030 0.70 KDM4E (0.36) KDM4EALDH1A1EGFRKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116057059-B Deuterated compounds useful as KRAS G12D inhibitors 南京燧坤智能科技有限公司 2024-03-08 CN disclosed
CN-116057059-A Deuterated compounds useful as KRAS G12D inhibitors 南京燧坤智能科技有限公司 2023-05-02 CN disclosed
WO-2023284881-A1 HETEROCYCLIC COMPOUNDS USEFUL AS KRAS G12D INHIBITORS SILEXON AI TECHNOLOGY CO., LTD. (CN) 2023-01-19 WO disclosed
WO-2022262838-A1 DEUTERATED COMPOUNDS USEFUL AS KRAS G12D INHIBITORS SILEXON AI TECHNOLOGY CO., LTD. (CN) 2022-12-22 WO disclosed