SCHEMBL29015696

SCHEMBL29015696

CS(=O)(=O)n1ccc2cccc(Nc3nc(Cl)ncc3F)c21

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GLO1 Q04760 3/20 0.43
AURKA O14965 9/20 0.39
AURKB Q96GD4 4/20 0.39
JAK2 O60674 2/20 0.35
ALK Q9UM73 2/20 0.34
SLC40A1 Q9NP59 1/20 0.34
ALDH1A1 P00352 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
SYK P43405 1/20 0.34
KMT2A Q03164 1/20 0.33
CDC7 O00311 1/20 0.33
MAPK8 P45983 1/20 0.33
CDK7 P50613 1/20 0.33
CDK9 P50750 1/20 0.33
GSK3A P49840 1/20 0.33
LRRK2 Q5S007 1/20 0.33
MAPK15 Q8TD08 1/20 0.33
CAMKK2 Q96RR4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30872003 1.00 GLO1 (0.43) GLO1AURKAAURKBJAK2ALK
SCHEMBL27238032 0.89 ALK (0.45) ALKCDK7CDK9
SCHEMBL30426111 0.89 ALK (0.45) ALKCDK7CDK9
SCHEMBL29015706 0.88 ALK (0.35) GLO1AURKAALKSLC40A1L3MBTL1
SCHEMBL30872014 0.88 ALK (0.35) GLO1AURKAALKSLC40A1L3MBTL1
SCHEMBL30424889 0.87 ALK (0.41) JAK2ALKSYKKMT2ACDC7
SCHEMBL29015730 0.87 ALK (0.41) JAK2ALKSYKKMT2ACDC7
SCHEMBL29216425 0.86 ULK1 (0.42) AURKBALKCDC7CDK7CDK9
SCHEMBL30871971 0.86 ULK1 (0.42) AURKBALKCDC7CDK7CDK9
Trifluoroacetic Acid SCHEMBL30730912 0.81 ALK (0.36) JAK2ALKSYKKMT2ACDC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117794914-A Pyrimidine-2, 4-diamine derivatives, process for preparing the same, and pharmaceutical composition for preventing or treating cancer comprising the same as active ingredient 韩国化学研究院 2024-03-29 CN disclosed
CN-116249690-A Indoline compounds and derivatives as EGFR inhibitors 百济神州有限公司 2023-06-09 CN disclosed