SCHEMBL29017308

SCHEMBL29017308

Cc1cccc(C)c1Nc1nc(Nc2ccc(N3CCOCC3)cc2)nc2[nH]ccc12.N[SH](=O)=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 1/20 0.53
BTK Q06187 1/20 0.53
TTK P33981 7/20 0.52
PTK2 Q05397 8/20 0.52
TTBK1 Q5TCY1 1/20 0.52
TTBK2 Q6IQ55 1/20 0.52
JAK2 O60674 1/20 0.50
BRD4 O60885 1/20 0.50
PIK3CB P42338 1/20 0.47
MAPK8 P45983 1/20 0.47
TP53 P04637 1/20 0.47
MAPT P10636 1/20 0.47
MAPK1 P28482 1/20 0.47
IGF1R P08069 1/20 0.46
CCNK O75909 1/20 0.46
CCNA2 P20248 1/20 0.46
CDK2 P24941 1/20 0.46
CCND3 P30281 1/20 0.46
CDK9 P50750 1/20 0.46
CDK6 Q00534 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29017291 0.90 PTK2 (0.54) TTKPTK2PIK3CBMAPK8IGF1R
SCHEMBL14547750 0.80 TTK (0.63) JAK3BTKTTKPTK2TTBK1
SCHEMBL29017299 0.79 CCND3 (0.52) JAK3BTKPTK2JAK2BRD4
SCHEMBL29017419 0.79 MAP4K1 (0.51) JAK3BTK
SCHEMBL4383026 0.78 JAK3 (0.59) JAK3BTKTTKPTK2TTBK1
SCHEMBL12085313 0.78 JAK3 (0.70) JAK3BTKTTKPTK2TTBK1
SCHEMBL4383739 0.78 JAK2 (0.60) JAK3BTKTTKPTK2TTBK1
SCHEMBL12085388 0.76 JAK3 (0.73) JAK3BTKTTKPTK2TTBK1
SCHEMBL24243309 0.76 TTK (0.67) JAK3BTKTTKPTK2TTBK1
SCHEMBL27806139 0.76 ZAP70 (0.72) TTBK1TTBK2JAK2TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116239597-A Pyrimidine pyrrole derivative and medicinal composition and application thereof 中国科学院上海药物研究所 2023-06-09 CN disclosed