SCHEMBL29017291

SCHEMBL29017291

Cc1cc(N2CCOCC2)ccc1Nc1nc(Nc2c(C)cccc2C)c2cc[nH]c2n1.N[SH](=O)=O

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTK2 Q05397 7/20 0.54
TTK P33981 13/20 0.54
PIK3CB P42338 1/20 0.54
MAPK8 P45983 1/20 0.54
IGF1R P08069 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29017308 0.90 JAK3 (0.53) PTK2TTKPIK3CBMAPK8IGF1R
SCHEMBL12429374 0.82 PTK2 (0.69) PTK2TTKMAPK8IGF1R
SCHEMBL29017290 0.79 TTK (0.65) PTK2TTKPIK3CBMAPK8IGF1R
SCHEMBL18696331 0.77 TTK (0.63) PTK2TTKIGF1R
SCHEMBL29017299 0.76 CCND3 (0.52) PTK2
SCHEMBL18696334 0.75 IGF1R (0.57) PTK2TTKPIK3CBMAPK8IGF1R
SCHEMBL18696330 0.72 ALK (0.65) PTK2TTKIGF1R
SCHEMBL12429379 0.72 PTK2 (0.85) PTK2TTKPIK3CBMAPK8IGF1R
SCHEMBL17731732 0.70 TTK (1.00) PTK2TTKPIK3CBMAPK8IGF1R
SCHEMBL4383739 0.70 JAK2 (0.60) PTK2TTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116239597-A Pyrimidine pyrrole derivative and medicinal composition and application thereof 中国科学院上海药物研究所 2023-06-09 CN claimed
CN-116239597-A Pyrimidine pyrrole derivative and medicinal composition and application thereof 中国科学院上海药物研究所 2023-06-09 CN disclosed