SCHEMBL29017299

SCHEMBL29017299

Cc1cccc(C)c1Nc1nc(Nc2ccc(N3CCN(C)CC3)cn2)nc2[nH]ccc12.N[SH](=O)=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCND3 P30281 11/20 0.52
CDK6 Q00534 11/20 0.52
CDK9 P50750 9/20 0.50
CCNK O75909 8/20 0.50
PTK2 Q05397 1/20 0.48
JAK2 O60674 1/20 0.47
BRD4 O60885 1/20 0.47
CTSC P53634 3/20 0.46
MAP4K1 Q92918 3/20 0.46
CCNT1 O60563 2/20 0.45
CDK4 P11802 1/20 0.45
CCND1 P24385 1/20 0.45
CDK7 P50613 1/20 0.45
CCNH P51946 1/20 0.45
MNAT1 P51948 1/20 0.45
CDK5 Q00535 1/20 0.45
CDK5R1 Q15078 1/20 0.45
CYP3A4 P08684 2/20 0.44
CCNA2 P20248 1/20 0.43
CDK2 P24941 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29017308 0.79 JAK3 (0.53) CCND3CDK6CDK9CCNKPTK2
SCHEMBL24327576 0.77 PTK2 (0.51) CCND3CDK6CDK9CCNKPTK2
SCHEMBL29017291 0.76 PTK2 (0.54) PTK2
SCHEMBL30372483 0.76 AXL (0.58) CCND3CDK6CDK9CCNKPTK2
SCHEMBL29017297 0.76 AXL (0.58) CCND3CDK6CDK9CCNKPTK2
SCHEMBL30736077 0.76 EGFR (0.66) CCND3CDK6CDK9CCNKPTK2
SCHEMBL23567021 0.76 EGFR (0.66) CCND3CDK6CDK9CCNKPTK2
SCHEMBL18696331 0.71 TTK (0.63) CCND3CDK6CDK9CCNKPTK2
SCHEMBL24327431 0.71 ALK (0.53) CCND3CDK6CDK9CCNKPTK2
SCHEMBL29015721 0.71 ALK (0.53) CCND3CDK6CDK9CCNKPTK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116239597-A Pyrimidine pyrrole derivative and medicinal composition and application thereof 中国科学院上海药物研究所 2023-06-09 CN disclosed