SCHEMBL29017698

SCHEMBL29017698

Nc1ccccc1-c1ccc(N2CCCC(NC(=O)c3ccc(Cl)c(Cl)c3)C2)nn1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.44
AURKA O14965 1/20 0.42
PDPK1 O15530 1/20 0.42
AURKB Q96GD4 1/20 0.42
PPARD Q03181 1/20 0.42
PPARA Q07869 1/20 0.42
CNR2 P34972 3/20 0.41
CA12 O43570 2/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA4 P22748 2/20 0.39
CA7 P43166 2/20 0.39
CA9 Q16790 2/20 0.39
BTK Q06187 4/20 0.39
JAK3 P52333 1/20 0.39
F10 P00742 1/20 0.38
UTS2R Q9UKP6 1/20 0.38
CNR1 P21554 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29017665 0.92 KMT2A (0.44) KMT2AMEN1AURKAPDPK1AURKB
SCHEMBL29637924 0.92 PPARD (0.47) KMT2AMEN1AURKAPDPK1AURKB
SCHEMBL29017668 0.92 PPARD (0.47) KMT2AMEN1AURKAPDPK1AURKB
SCHEMBL29017722 0.90 CNR1 (0.46) KMT2AMEN1AURKAPDPK1AURKB
SCHEMBL29017684 0.88 KMT2A (0.43) KMT2AMEN1PPARDPPARABTK
SCHEMBL29637951 0.88 PPARA (0.44) KMT2AMEN1AURKAPDPK1AURKB
SCHEMBL29017740 0.88 PPARA (0.44) KMT2AMEN1AURKAPDPK1AURKB
SCHEMBL29637930 0.88 KMT2A (0.43) KMT2AMEN1PPARDPPARABTK
SCHEMBL29017680 0.87 CNR2 (0.45) KMT2AMEN1PPARDPPARACNR2
SCHEMBL29637950 0.87 CNR2 (0.45) KMT2AMEN1PPARDPPARACNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114478478-B N- (1- (6- (substituted phenyl) pyridazin-3-yl) piperidin-3-yl) amine/amide derivatives and process for preparing the same 厦门大学 2023-06-13 CN disclosed
CN-114478478-A N- (1- (6- (substituted phenyl) pyridazine-3-yl) piperidine-3-yl) amine/amide derivative and preparation method thereof 厦门大学 2022-05-13 CN disclosed