SCHEMBL29017665

SCHEMBL29017665

Nc1ccccc1-c1ccc(N2CCCC(NC(=O)c3ccc(Cl)c(F)c3)C2)nn1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
AURKA O14965 1/20 0.41
PDPK1 O15530 1/20 0.41
AURKB Q96GD4 1/20 0.41
F10 P00742 1/20 0.40
PPARD Q03181 1/20 0.40
PPARA Q07869 1/20 0.40
RORC P51449 1/20 0.39
CNR2 P34972 4/20 0.39
DGAT2 Q96PD7 1/20 0.39
BTK Q06187 3/20 0.38
S100A4 P26447 1/20 0.38
CDK7 P50613 1/20 0.38
JAK3 P52333 1/20 0.38
CNR1 P21554 1/20 0.37
ACKR3 P25106 1/20 0.37
PKM P14618 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29017698 0.92 KMT2A (0.44) KMT2AMEN1AURKAPDPK1AURKB
SCHEMBL29017746 0.92 KMT2A (0.46) KMT2AMEN1AURKAPDPK1AURKB
SCHEMBL29637977 0.92 KMT2A (0.46) KMT2AMEN1AURKAPDPK1AURKB
SCHEMBL29637895 0.89 PKM (0.43) KMT2AMEN1F10PPARDPPARA
SCHEMBL29017648 0.88 KMT2A (0.42) KMT2AMEN1AURKAPDPK1AURKB
SCHEMBL29017722 0.88 CNR1 (0.46) KMT2AMEN1AURKAPDPK1AURKB
SCHEMBL29017668 0.84 PPARD (0.47) KMT2AMEN1AURKAPDPK1AURKB
SCHEMBL29637924 0.84 PPARD (0.47) KMT2AMEN1AURKAPDPK1AURKB
SCHEMBL29017667 0.84 AURKA (0.44) KMT2AMEN1AURKAPDPK1AURKB
SCHEMBL29017647 0.82 BTK (0.52) BTKJAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114478478-B N- (1- (6- (substituted phenyl) pyridazin-3-yl) piperidin-3-yl) amine/amide derivatives and process for preparing the same 厦门大学 2023-06-13 CN disclosed
CN-114478478-A N- (1- (6- (substituted phenyl) pyridazine-3-yl) piperidine-3-yl) amine/amide derivative and preparation method thereof 厦门大学 2022-05-13 CN disclosed