SCHEMBL290195

SCHEMBL290195

Cc1nc(NCC(=O)c2ccc(-c3cc4ccccc4s3)s2)sc1C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 9/20 0.49
RAB9A P51151 8/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
ALDH1A1 P00352 2/20 0.40
PKM P14618 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
BCL2L1 Q07817 1/20 0.38
PDE5A O76074 1/20 0.37
PDE1A P54750 1/20 0.37
PDE1B Q01064 1/20 0.37
PDE1C Q14123 1/20 0.37
MAPT P10636 3/20 0.36
HPGD P15428 2/20 0.36
DHODH Q02127 2/20 0.36
POLB P06746 1/20 0.36
TSHR P16473 1/20 0.36
RPS6KB2 Q9UBS0 1/20 0.36
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL290238 0.76 SMN1; SMN2 (0.56) NPC1RAB9ASMN1; SMN2ALDH1A1BCL2L1
SCHEMBL290196 0.75 SMN1; SMN2 (0.40) NPC1RAB9ASMN1; SMN2BCL2L1RPS6KB2
SCHEMBL289628 0.74 SMN1; SMN2 (0.63) NPC1RAB9ASMN1; SMN2ALDH1A1PKM
SCHEMBL6412727 0.73 BCL2L1 (0.64) RAB9AALDH1A1BCL2L1HPGDPOLB
SCHEMBL289881 0.72 SMN1; SMN2 (0.61) NPC1RAB9ASMN1; SMN2ALDH1A1BCL2L1
SCHEMBL290152 0.69 SMN1; SMN2 (0.53) NPC1RAB9ASMN1; SMN2ALDH1A1BCL2L1
SCHEMBL290016 0.69 SMN1; SMN2 (0.56) NPC1RAB9ASMN1; SMN2ALDH1A1BCL2L1
SCHEMBL289595 0.69 SMN1; SMN2 (0.68) NPC1RAB9ASMN1; SMN2ALDH1A1MAPT
SCHEMBL4919866 0.69 NPC1 (0.75) NPC1RAB9ASMN1; SMN2ALDH1A1PKM
Hydrochloric Acid SCHEMBL8555706 0.68 NPC1 (0.73) NPC1RAB9ASMN1; SMN2ALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427447-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION Pike Pharma GmbH (CH) 2012-03-14 EP disclosed
WO-2010128163-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION PIKE PHARMA GMBH (CH) 2010-11-11 WO disclosed