SCHEMBL29020109

SCHEMBL29020109

Cn1cc(-c2nc(C(=O)O)cc(-c3ccnc(F)c3)n2)cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.44
STING1 Q86WV6 1/20 0.41
CLK2 P49760 1/20 0.40
LRRK2 Q5S007 1/20 0.40
MAP4K4 O95819 1/20 0.40
CCNC P24863 1/20 0.39
CDK8 P49336 1/20 0.39
PIM1 P11309 1/20 0.39
PIM2 Q9P1W9 1/20 0.39
MAP3K12 Q12852 1/20 0.39
IDO1 P14902 1/20 0.39
SYK P43405 1/20 0.38
GRM2 Q14416 1/20 0.38
FGFR1 P11362 2/20 0.37
FGFR2 P21802 2/20 0.37
FGFR3 P22607 2/20 0.37
FGFR4 P22455 1/20 0.37
KDR P35968 1/20 0.37
MKNK1 Q9BUB5 2/20 0.37
EGFR P00533 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29020164 0.85 CHEK1 (0.57) CHEK1STING1CLK2LRRK2MAP4K4
SCHEMBL29961571 0.85 CHEK1 (0.57) CHEK1STING1CLK2LRRK2MAP4K4
SCHEMBL29961693 0.83 CHEK1 (0.53) CHEK1STING1MAP4K4CCNCCDK8
SCHEMBL29020112 0.83 CHEK1 (0.53) CHEK1STING1MAP4K4CCNCCDK8
SCHEMBL29020185 0.82 ROCK2 (0.47) CLK2LRRK2EGFR
SCHEMBL29020125 0.79 CHEK1 (0.53) CHEK1MAP4K4CCNCCDK8PIM1
SCHEMBL29020180 0.78 CHEK1 (0.50) CHEK1MAP4K4CCNCCDK8PIM1
SCHEMBL29961338 0.78 CHEK1 (0.50) CHEK1MAP4K4CCNCCDK8PIM1
SCHEMBL29961343 0.78 CLK2 (0.56) CHEK1CLK2LRRK2MAP4K4CCNC
SCHEMBL31174355 0.78 CHEK1 (0.47) CHEK1STING1CLK2LRRK2MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115093400-B AhR inhibitor, application and preparation method thereof 北京华森英诺生物科技有限公司 2023-09-05 CN disclosed
CN-115093400-A AhR inhibitor and application and preparation method thereof 重庆华森制药股份有限公司 2022-09-23 CN disclosed