SCHEMBL29020185

SCHEMBL29020185

CC(NC(=O)c1cc(-c2ccnc(F)c2)nc(-c2cnn(C)c2)n1)c1ccnc(F)c1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.47
PRKG1 Q13976 3/20 0.47
PRKACA P17612 2/20 0.47
PRKACG P22612 2/20 0.47
PRKACB P22694 2/20 0.47
AKT1 P31749 2/20 0.47
CYP2C9 P11712 1/20 0.44
ROCK1 Q13464 1/20 0.44
KCNT1 Q5JUK3 1/20 0.41
CLK1 P49759 5/20 0.40
MAPK1 P28482 4/20 0.39
PFKFB3 Q16875 1/20 0.39
EGFR P00533 1/20 0.39
CLK2 P49760 1/20 0.39
LRRK2 Q5S007 1/20 0.39
RAB9A P51151 1/20 0.39
MET P08581 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29020117 0.96 KCNT1 (0.44) ROCK2PRKG1PRKACAPRKACGPRKACB
SCHEMBL29020149 0.93 MAPK1 (0.44) ROCK2PRKG1PRKACAPRKACGPRKACB
SCHEMBL29020210 0.91 CLK1 (0.48) ROCK2PRKG1PRKACAPRKACGPRKACB
SCHEMBL29020227 0.90 PDE2A (0.43) ROCK2PRKG1PRKACAPRKACGPRKACB
SCHEMBL29020203 0.89 PHGDH (0.41) ROCK2PRKG1PRKACAPRKACGPRKACB
SCHEMBL29020173 0.87 AHR (0.51) ROCK2PRKG1PRKACAPRKACGPRKACB
SCHEMBL29020109 0.82 CHEK1 (0.44) EGFRCLK2LRRK2
SCHEMBL29020122 0.82 MAPK1 (0.49) ROCK2ROCK1KCNT1CLK1MAPK1
SCHEMBL29020127 0.82 MAPK1 (0.49) ROCK2ROCK1KCNT1CLK1MAPK1
SCHEMBL29961598 0.82 MAPK1 (0.49) ROCK2ROCK1KCNT1CLK1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115093400-B AhR inhibitor, application and preparation method thereof 北京华森英诺生物科技有限公司 2023-09-05 CN disclosed
CN-115093400-A AhR inhibitor and application and preparation method thereof 重庆华森制药股份有限公司 2022-09-23 CN disclosed