Asparagine

Asparagine

SCHEMBL2902050

CC(C)[C@H](N)C(N)=O.C[C@H](N)C(=O)O.NC(=O)C[C@H](N)C(=O)O.O=C(O)[C@H]1NCC[C@@H]1c1ccc2ccccc2c1

nearest known ligand 0.39

Full drug profile on Sugi Atlas →

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SLC1A3 P43003 1/20 0.34
SLC1A2 P43004 1/20 0.34
SLC1A1 P43005 1/20 0.34
TPH1 P17752 1/20 0.33
EPHX1 P07099 1/20 0.32
MC4R P32245 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Asparagine SCHEMBL2927424 0.79 SLC1A3 (0.32) SLC1A3SLC1A2SLC1A1
SCHEMBL13125707 0.77 SLC6A4 (0.44)
Asparagine SCHEMBL2902137 0.76 MC4R (0.35) MC4R
Asparagine SCHEMBL7855644 0.73 SLC1A3 (0.34) SLC1A3SLC1A2SLC1A1TPH1
Leucine SCHEMBL7627315 0.72 SLC7A5 (0.44) SLC1A3SLC1A2MC4R
Asparagine SCHEMBL7855451 0.69 MC4R (0.36) MC4R
Leucine SCHEMBL2299788 0.69 SLC7A5 (0.40) MC4R
SCHEMBL2903921 0.67 SLC6A4 (0.55)
SCHEMBL7356872 0.67 SLC6A4 (0.55)
Asparagine SCHEMBL8942998 0.65 GRIK1 (0.41) SLC1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2239270-A2 Low molecular weight peptide derivatives as inhibitors of the Laminin/Nidogen interaction Sanofi-Aventis Deutschland GmbH (DE) 2010-10-13 EP disclosed
EP-1845106-B1 Low molecular weight peptide derivatives as inhibitors of the laminin/nidogen interaction SANOFI AVENTIS DEUTSCHLAND (DE) 2010-08-11 EP disclosed
EP-1845106-A1 Low molecular weight peptide derivatives as inhibitors of the laminin/nidogen interaction Sanofi-Aventis Deutschland GmbH (DE) 2007-10-17 EP disclosed
EP-1157040-B1 LOW MOLECULAR WEIGHT PEPTIDE DERIVATIVES AS INHIBITORS OF THE LAMININ/NIDOGEN INTERACTION SANOFI AVENTIS DEUTSCHLAND (DE) 2007-08-22 EP disclosed
US-6365572-B1 FOR THERAPY OF DISEASES RELATED TO INCREASED OR UNWANTED SYNTHESIS OF BASEMENT MEMBRANES SUCH AS DIABETES MELLITUS; ATHEROSCLEROSIS; CANCER; DIABETIC RETINOPATHIA; FIBROPLASIA RETROLENTALIS; OR PSORIASIS, RHEUMATOIC ARTHRITIS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2002-04-02 US disclosed
EP-1157040-A1 LOW MOLECULAR WEIGHT PEPTIDE DERIVATIVES AS INHIBITORS OF THE LAMININ/NIDOGEN INTERACTION Aventis Pharma Deutschland GmbH (DE) 2001-11-28 EP disclosed
EP-1070727-A1 Low molecular weight peptide derivatives as inhibitors of the laminin/nidogen interaction Aventis Pharma Deutschland GmbH (DE) 2001-01-24 EP disclosed
WO-2000052051-A1 LOW MOLECULAR WEIGHT PEPTIDE DERIVATIVES AS INHIBITORS OF THE LAMININ/NIDOGEN INTERACTION AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-09-08 WO disclosed