SCHEMBL29020535

SCHEMBL29020535

Fc1ccc(CSc2nnc(-c3ccc(F)cc3)n2-c2ccc(I)cc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TERT O14746 2/20 0.58
METAP2 P50579 2/20 0.57
PTGS2 P35354 1/20 0.55
MEN1 O00255 3/20 0.52
KMT2A Q03164 3/20 0.52
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51
LMNA P02545 2/20 0.49
ALDH1A1 P00352 2/20 0.49
NPSR1 Q6W5P4 1/20 0.49
SMN1; SMN2 Q16637 3/20 0.48
PTK2 Q05397 2/20 0.47
CRHBP P24387 1/20 0.46
HTT P42858 1/20 0.46
CRHR2 Q13324 1/20 0.46
GAA P10253 1/20 0.46
HPGD P15428 1/20 0.46
MAPK1 P28482 1/20 0.46
HDAC3 O15379 1/20 0.45
HDAC1 Q13547 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29020514 0.92 CYP3A4 (0.53) TERTMETAP2PTGS2MEN1KMT2A
SCHEMBL29020512 0.91 CYP3A4 (0.57) TERTMETAP2PTGS2MEN1KMT2A
SCHEMBL30498867 0.88 METAP2 (0.52) TERTMETAP2PTGS2MEN1KMT2A
SCHEMBL29020511 0.88 METAP2 (0.52) TERTMETAP2PTGS2MEN1KMT2A
SCHEMBL29020560 0.83 PTK2 (0.54) TERTMETAP2PTGS2MEN1KMT2A
SCHEMBL6404838 0.80 CYP3A4 (0.78) TERTMETAP2PTGS2MEN1KMT2A
SCHEMBL28376474 0.76 MAPK1 (0.54) TERTMETAP2PTGS2MEN1KMT2A
SCHEMBL16486457 0.75 PTK2 (0.61) TERTMETAP2PTGS2MEN1KMT2A
SCHEMBL28372567 0.74 SMN1; SMN2 (0.53) TERTMETAP2PTGS2MEN1KMT2A
SCHEMBL28376596 0.73 MEN1 (0.55) TERTMETAP2MEN1KMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113402473-B Thiotriazole compound, preparation method and application thereof 四川省医学科学院·四川省人民医院 2023-06-23 CN disclosed
CN-113402473-A Thiotriazole compound, preparation method and application thereof 四川省医学科学院·四川省人民医院 2021-09-17 CN disclosed