SCHEMBL29021864

SCHEMBL29021864

COC(=O)c1c([N+](=O)[O-])ccc(Oc2c(F)ccc(N)c2Cl)c1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.41
ALDH1A1 P00352 3/20 0.38
MAPT P10636 7/20 0.36
POLB P06746 3/20 0.36
KMT2A Q03164 7/20 0.36
SETD7 Q8WTS6 1/20 0.36
LMNA P02545 3/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
MEN1 O00255 5/20 0.35
KDM4E B2RXH2 2/20 0.35
ALOX12 P18054 2/20 0.35
TTR P02766 1/20 0.35
ALB P02768 1/20 0.35
THRB P10828 1/20 0.35
MAPK1 P28482 2/20 0.35
ABCC4 O15439 1/20 0.35
PLIN1 O60240 1/20 0.35
CACNA1F O60840 1/20 0.35
GMNN O75496 1/20 0.35
KCNK2 O95069 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30353744 1.00 TDP1 (0.41) TDP1ALDH1A1MAPTPOLBKMT2A
SCHEMBL29021770 0.92 TDP1 (0.42) TDP1ALDH1A1MAPTPOLBKMT2A
SCHEMBL30353742 0.92 TDP1 (0.42) TDP1ALDH1A1MAPTPOLBKMT2A
SCHEMBL29021594 0.91 TDP1 (0.41) TDP1ALDH1A1MAPTPOLBKMT2A
SCHEMBL30353743 0.91 TDP1 (0.41) TDP1ALDH1A1MAPTPOLBKMT2A
SCHEMBL30396199 0.89 KMT2A (0.39) TDP1MAPTPOLBKMT2ALMNA
SCHEMBL29561773 0.89 LMNA (0.36) TDP1ALDH1A1MAPTPOLBKMT2A
SCHEMBL22832028 0.89 LMNA (0.36) TDP1ALDH1A1MAPTPOLBKMT2A
SCHEMBL29021712 0.80 TDP1 (0.36) TDP1ALDH1A1MAPTPOLBKMT2A
SCHEMBL30353776 0.80 TDP1 (0.36) TDP1ALDH1A1MAPTPOLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116096710-A 4-oxo-3, 4-dihydroquinazolinone compounds for the treatment of BRAF related diseases and disorders 阿雷生物药品公司 2023-05-09 CN disclosed