SCHEMBL29026149

SCHEMBL29026149

NC(=O)c1nc(C(F)(F)F)ccc1-c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.43
MAP2K3 P46734 1/20 0.43
BCAT2 O15382 2/20 0.42
IKBKB O14920 1/20 0.42
PDE4B Q07343 2/20 0.40
SYK P43405 2/20 0.40
IDH2 P48735 1/20 0.40
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
KDM4E B2RXH2 3/20 0.40
HSD17B10 Q99714 2/20 0.40
ADORA2A P29274 1/20 0.40
LMNA P02545 2/20 0.39
POLB P06746 1/20 0.39
PDE11A Q9HCR9 1/20 0.39
PDE10A Q9Y233 1/20 0.39
HPGD P15428 2/20 0.39
ALDH1A1 P00352 1/20 0.39
TSHR P16473 1/20 0.39
P2RX7 Q99572 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29800136 0.85 IKBKB (0.44) IKBKBPDE4BPTGS1PTGS2LMNA
SCHEMBL945449 0.80 HSP90AA1 (0.52) PTGS1PTGS2
SCHEMBL30627185 0.80 F2 (0.42) IKBKBIDH2PTGS1PTGS2KDM4E
SCHEMBL59061 0.78 JAK2 (0.41) JAK2BCAT2SYKIDH2PTGS1
SCHEMBL27896613 0.77 MAP2K3 (0.51) MAP2K3BCAT2IKBKBKDM4EHSD17B10
SCHEMBL31374321 0.77 PDE4B (0.38) PDE4BSYKADORA2APDE11APDE10A
SCHEMBL27651135 0.76 MAP2K3 (0.46) MAP2K3BCAT2IKBKBKDM4EHSD17B10
SCHEMBL4504523 0.75 JAK2 (0.49) JAK2BCAT2KDM4EHSD17B10LMNA
SCHEMBL2159117 0.75 MAP2K3 (0.49) JAK2MAP2K3IKBKBPDE4BSYK
SCHEMBL30627079 0.74 TRPA1 (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116348115-A Combination of antibody-drug conjugate and PARP1 selective inhibitor 阿斯利康(英国)有限公司 2023-06-27 CN disclosed