SCHEMBL2903516

SCHEMBL2903516

O=C(NCC(O)c1ccccc1)Oc1ccc2cc(-c3n[nH]c4ccsc34)[nH]c2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITK Q08881 18/20 0.47
LCK P06239 3/20 0.47
TXK P42681 3/20 0.47
SYK P43405 3/20 0.47
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
PLK4 O00444 1/20 0.37
CHEK1 O14757 1/20 0.37
AURKA O14965 1/20 0.37
CCNB2 O95067 1/20 0.37
ABL1 P00519 1/20 0.37
CDK1 P06493 1/20 0.37
PDGFRB P09619 1/20 0.37
CDK4 P11802 1/20 0.37
SRC P12931 1/20 0.37
CCNB1 P14635 1/20 0.37
CCNA2 P20248 1/20 0.37
CCND1 P24385 1/20 0.37
CDK2 P24941 1/20 0.37
WEE1 P30291 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1621145 0.85 ITK (0.54) ITKLCKTXKSYKNPC1
SCHEMBL2898022 0.80 ITK (0.47) ITKLCKTXKSYKNPC1
SCHEMBL2898497 0.80 ITK (0.59) ITKLCKTXKSYKPLK4
SCHEMBL27645971 0.79 ITK (0.62) ITKLCKTXKSYKPLK4
SCHEMBL2898574 0.78 ITK (0.45) ITKLCKTXKSYKNPC1
SCHEMBL2902831 0.76 ITK (0.45) ITKLCKTXKSYKNPC1
SCHEMBL2903568 0.73 ITK (0.43) ITKLCKTXKSYKNPC1
SCHEMBL1621146 0.71 ITK (0.48) ITKLCKTXKSYKKDR
SCHEMBL1623341 0.71 ITK (0.63) ITKLCKTXKSYK
SCHEMBL13869803 0.71 ITK (0.60) ITKLCKTXKSYKNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682553-B1 THIENOPYRAZOLES AVENTIS PHARMA INC (US) 2010-05-19 EP claimed