SCHEMBL29030308

SCHEMBL29030308

Cc1ccc(-c2c(C(=O)O)[nH]c3cccnc23)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE9A O76083 1/20 0.56
ALDH1A1 P00352 4/20 0.53
KDM4E B2RXH2 3/20 0.53
HPGD P15428 3/20 0.53
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
HTT P42858 1/20 0.53
GFER P55789 1/20 0.53
HSD17B10 Q99714 1/20 0.53
TGFBR1 P36897 3/20 0.43
MAPK14 Q16539 1/20 0.42
MAP2 P11137 1/20 0.41
MCL1 Q07820 2/20 0.41
GAA P10253 2/20 0.40
GLA P06280 1/20 0.40
GSK3B P49841 1/20 0.40
ADK P55263 1/20 0.40
GPR35 Q9HC97 3/20 0.40
COMT P21964 1/20 0.40
RPA1 P27694 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18322288 0.86 MAP2 (0.53) PDE9AALDH1A1KDM4EHPGDMEN1
SCHEMBL18322246 0.83 PDE9A (0.51) PDE9AALDH1A1KDM4EHPGDMEN1
SCHEMBL5264870 0.82 MAPT (0.57) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL5264866 0.82 MAPT (0.57) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL27523327 0.80 HPGD (0.50) PDE9AALDH1A1KDM4EHPGDMEN1
SCHEMBL3883122 0.80 HPSE (0.50) PDE9AKDM4ETGFBR1SMN1; SMN2
SCHEMBL22907746 0.77 MAP2 (0.53) PDE9ATGFBR1MAPK14MAP2GAA
SCHEMBL3877998 0.75 PARP1 (0.48) PDE9AMAPK14MAP2
SCHEMBL27791164 0.74 DHODH (0.50) ALDH1A1KDM4EHPGDMAPK14
SCHEMBL21292084 0.74 TGFBR1 (0.44) PDE9AALDH1A1KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107787322-B Tricyclic compounds and their use as phosphodiesterase inhibitors 辉瑞大药厂 2023-07-07 CN disclosed