SCHEMBL29030508

SCHEMBL29030508

CCOCOc1cc(C)cc(C)c1-c1cnc(N[C@@H]2CCCN(C(=O)O)C2)nn1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IL1B P01584 1/20 0.37
NLRP3 Q96P20 1/20 0.37
JAK3 P52333 2/20 0.36
EGFR P00533 1/20 0.36
ITK Q08881 1/20 0.36
CCNK O75909 7/20 0.35
CCNA2 P20248 7/20 0.35
CDK2 P24941 7/20 0.35
CDK7 P50613 7/20 0.35
CCNH P51946 7/20 0.35
MNAT1 P51948 7/20 0.35
CDK12 Q9NYV4 7/20 0.35
JAK1 P23458 1/20 0.34
GFER P55789 3/20 0.34
MAPK8 P45983 2/20 0.34
MAPK9 P45984 2/20 0.34
GSK3B P49841 2/20 0.34
MAPK10 P53779 2/20 0.34
MAPK14 Q16539 2/20 0.34
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29030511 1.00 IL1B (0.37) IL1BNLRP3JAK3EGFRITK
SCHEMBL29030479 0.90 BTK (0.39) IL1BNLRP3JAK3JAK1
SCHEMBL29030478 0.90 BTK (0.39) IL1BNLRP3JAK3JAK1
SCHEMBL30488543 0.90 BTK (0.39) IL1BNLRP3JAK3JAK1
SCHEMBL29042803 0.89 NLRP3 (0.37) IL1BNLRP3
SCHEMBL26092921 0.87 IL1B (0.47) IL1BNLRP3CCNKCDK2CDK12
SCHEMBL26092924 0.87 IL1B (0.47) IL1BNLRP3CCNKCDK2CDK12
SCHEMBL29042799 0.86 NLRP3 (0.37) IL1BNLRP3JAK3CDK2JAK1
SCHEMBL29042800 0.86 NLRP3 (0.37) IL1BNLRP3JAK3CDK2JAK1
SCHEMBL26439664 0.86 PIK3CD (0.39) IL1BNLRP3JAK3JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116410140-A NLRP3 inflammation corpuscle inhibitor and application thereof 药捷安康(南京)科技股份有限公司 2023-07-11 CN disclosed