SCHEMBL2903470

SCHEMBL2903470

CCOC(=O)CC1C(=O)N(CCCN2CCCCC2)CCN1C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.40
HRH3 Q9Y5N1 8/20 0.37
KCNH2 Q12809 1/20 0.36
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 3/20 0.36
KMT2A Q03164 1/20 0.35
CACNA1F O60840 1/20 0.34
BCHE P06276 1/20 0.34
CACNA1D Q01668 1/20 0.34
CACNA1S Q13698 1/20 0.34
CACNA1C Q13936 1/20 0.34
HRH4 Q9H3N8 1/20 0.34
CYP1A2 P05177 1/20 0.34
MAPK1 P28482 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1344381 0.86 POLB (0.37) POLBHRH3KCNH2KMT2A
SCHEMBL1344109 0.78 ACHE (0.42) BCHETDP1
SCHEMBL1344107 0.78 ACHE (0.42) BCHETDP1
SCHEMBL3170887 0.77 CYP1A2 (0.41) POLBHRH3ALDH1A1KDM4EKMT2A
SCHEMBL1569345 0.77 CYP1A2 (0.41) POLBHRH3ALDH1A1KDM4EKMT2A
SCHEMBL1344122 0.72 HRH3 (0.36) HRH3
SCHEMBL28337206 0.71 GSK3A (0.38) POLBALDH1A1KMT2ASMN1; SMN2TDP1
SCHEMBL28337208 0.71 GSK3A (0.38) POLBALDH1A1KMT2ASMN1; SMN2TDP1
SCHEMBL1344389 0.70 HRH3 (0.35) HRH3KMT2A
SCHEMBL1343917 0.70 HRH3 (0.35) HRH3KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2220055-A2 NOVEL HETEROCYCLYL COMPOUNDS AND THEIR USE AS CHEMOKINE ANTAGONISTS F. Hoffmann-La Roche AG (CH) 2010-08-25 EP disclosed
WO-2009010429-A2 NOVEL HETEROCYCLYL COMPOUNDS AND THEIR USE AS CHEMOKINE ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2009-01-22 WO disclosed