SCHEMBL2903702

SCHEMBL2903702

O=C(C=Cc1ccc(Cl)cc1Cl)N1CCC(=O)N(CCN2CCCC2)CC1

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.58
ALDH1A1 P00352 2/20 0.58
SMN1; SMN2 Q16637 5/20 0.50
GAA P10253 2/20 0.50
LMNA P02545 4/20 0.49
L3MBTL1 Q9Y468 2/20 0.49
MAPT P10636 4/20 0.45
NPC1 O15118 1/20 0.45
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
MAPK1 P28482 1/20 0.43
ITGB2 P05107 4/20 0.42
ICAM1 P05362 4/20 0.42
ITGAL P20701 4/20 0.42
GPR183 P32249 2/20 0.42
CCR1 P32246 1/20 0.41
NPSR1 Q6W5P4 1/20 0.40
F2R P25116 1/20 0.40
ENPP2 Q13822 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2903699 1.00 RAB9A (0.58) RAB9AALDH1A1SMN1; SMN2GAALMNA
SCHEMBL2905287 0.85 GAA (0.57) RAB9AALDH1A1GAALMNAL3MBTL1
SCHEMBL2905291 0.85 GAA (0.57) RAB9AALDH1A1GAALMNAL3MBTL1
SCHEMBL2904334 0.84 MEN1 (0.51) ALDH1A1GAALMNAL3MBTL1MAPT
SCHEMBL2904336 0.84 MEN1 (0.51) ALDH1A1GAALMNAL3MBTL1MAPT
SCHEMBL2903391 0.82 NPC1 (0.57) RAB9ANPC1GPR183
SCHEMBL2903396 0.82 NPC1 (0.57) RAB9ANPC1GPR183
SCHEMBL2905043 0.82 APP (0.47) RAB9AALDH1A1LMNAITGALGPR183
SCHEMBL2905040 0.82 APP (0.47) RAB9AALDH1A1LMNAITGALGPR183
SCHEMBL2897317 0.82 NPC1 (0.56) RAB9ANPC1GPR183

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010506-B1 DIAZEPAN DERIVATIVES MODULATORS OF CHEMOKINE RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-04 EP disclosed