SCHEMBL2905040

SCHEMBL2905040

O=C(/C=C/c1ccc(F)cc1F)N1CCC(=O)N(CCN2CCCC2)CC1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.47
GPR183 P32249 3/20 0.45
HRH3 Q9Y5N1 1/20 0.42
ALDH1A1 P00352 3/20 0.42
LMNA P02545 1/20 0.41
TP53 P04637 1/20 0.41
F2R P25116 1/20 0.40
ADRA1B P35368 1/20 0.40
CCR1 P32246 1/20 0.39
ITGAL P20701 1/20 0.39
CCNC P24863 1/20 0.39
CDK8 P49336 1/20 0.39
RAB9A P51151 1/20 0.39
DRD2 P14416 2/20 0.38
DRD3 P35462 2/20 0.38
PARP1 P09874 1/20 0.38
PELI1 Q96FA3 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2905043 1.00 APP (0.47) APPGPR183HRH3ALDH1A1LMNA
SCHEMBL2902873 0.85 ALDH1A1 (0.60) GPR183ALDH1A1LMNATP53RAB9A
SCHEMBL2902877 0.85 ALDH1A1 (0.60) GPR183ALDH1A1LMNATP53RAB9A
SCHEMBL2898842 0.84 L3MBTL1 (0.53) GPR183HRH3ALDH1A1LMNATP53
SCHEMBL2898840 0.84 L3MBTL1 (0.53) GPR183HRH3ALDH1A1LMNATP53
SCHEMBL2904962 0.83 GPR183 (0.45) GPR183HRH3ALDH1A1LMNATP53
SCHEMBL2904959 0.83 GPR183 (0.45) GPR183HRH3ALDH1A1LMNATP53
SCHEMBL2903699 0.82 RAB9A (0.58) GPR183ALDH1A1LMNAF2RCCR1
SCHEMBL2903702 0.82 RAB9A (0.58) GPR183ALDH1A1LMNAF2RCCR1
SCHEMBL2904919 0.79 HPGD (0.65) ALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010506-B1 DIAZEPAN DERIVATIVES MODULATORS OF CHEMOKINE RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-04 EP disclosed