SCHEMBL29039428

SCHEMBL29039428

CC(=O)Nc1nc(-c2ccc(F)cc2)c(-c2ccnc(Cl)n2)s1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.58
EGFR P00533 3/20 0.53
ALDH1A1 P00352 3/20 0.52
MAPT P10636 2/20 0.52
KDM4E B2RXH2 1/20 0.52
LMNA P02545 1/20 0.52
GAA P10253 1/20 0.52
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
PIK3CA P42336 3/20 0.48
MTOR P42345 1/20 0.46
PIK3CD O00329 1/20 0.46
PIK3CG P48736 1/20 0.46
PIK3C3 Q8NEB9 1/20 0.46
PKM P14618 1/20 0.46
DYRK1A Q13627 2/20 0.45
ADORA2A P29274 3/20 0.43
ADORA1 P30542 2/20 0.43
PDPK1 O15530 1/20 0.43
GRM5 P41594 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30410499 1.00 KCNH2 (0.58) KCNH2EGFRALDH1A1MAPTKDM4E
SCHEMBL30409799 0.84 EGFR (0.49) KCNH2EGFRALDH1A1MAPTKDM4E
SCHEMBL29039434 0.84 EGFR (0.49) KCNH2EGFRALDH1A1MAPTKDM4E
SCHEMBL30409188 0.82 EGFR (0.60) KCNH2EGFR
SCHEMBL29039435 0.82 EGFR (0.60) KCNH2EGFR
SCHEMBL30409186 0.82 EGFR (0.53) EGFR
SCHEMBL29039270 0.82 EGFR (0.53) EGFR
SCHEMBL1641694 0.80 BRAF (0.49) KCNH2EGFRALDH1A1MAPTGAA
SCHEMBL29039452 0.80 EGFR (0.52) EGFRALDH1A1KDM4EGAAKMT2A
SCHEMBL29039439 0.78 PTGS2 (0.51) KCNH2EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116143773-B 2-amino-4-thiazolylpyrimidine compound and preparation method and application thereof 中国药科大学 2023-07-21 CN disclosed
CN-116143773-A 2-amino-4-thiazolylpyrimidine compound and preparation method and application thereof 中国药科大学 2023-05-23 CN disclosed