SCHEMBL29039434

SCHEMBL29039434

CNc1nc(-c2ccc(F)cc2)c(-c2ccnc(Cl)n2)s1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.49
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
MAPT P10636 1/20 0.47
CCNT1 O60563 1/20 0.43
CDK9 P50750 1/20 0.43
KCNH2 Q12809 5/20 0.42
ACHE P22303 1/20 0.41
TGFBR1 P36897 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30409799 1.00 EGFR (0.49) EGFRKDM4EALDH1A1MAPTCCNT1
SCHEMBL29039270 0.84 EGFR (0.53) EGFR
SCHEMBL30409186 0.84 EGFR (0.53) EGFR
SCHEMBL29039452 0.84 EGFR (0.52) EGFRKDM4EALDH1A1
SCHEMBL30410176 0.84 EGFR (0.52) EGFRKDM4EALDH1A1
SCHEMBL30410499 0.84 KCNH2 (0.58) EGFRKDM4EALDH1A1MAPTKCNH2
SCHEMBL29039428 0.84 KCNH2 (0.58) EGFRKDM4EALDH1A1MAPTKCNH2
SCHEMBL29039439 0.83 PTGS2 (0.51) EGFRKCNH2ACHETGFBR1
SCHEMBL30410597 0.83 PTGS2 (0.51) EGFRKCNH2ACHETGFBR1
SCHEMBL5822178 0.82 EGFR (0.46) EGFRKDM4EALDH1A1MAPTCCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116143773-B 2-amino-4-thiazolylpyrimidine compound and preparation method and application thereof 中国药科大学 2023-07-21 CN disclosed
CN-116143773-A 2-amino-4-thiazolylpyrimidine compound and preparation method and application thereof 中国药科大学 2023-05-23 CN disclosed