SCHEMBL29040344

SCHEMBL29040344

Cc1nn(C)c2cc(C(N)=NO)cnc12

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA2B P29275 1/20 0.35
BRAF P15056 1/20 0.33
MAPK3 P27361 1/20 0.33
MAPK1 P28482 1/20 0.33
NTRK1 P04629 2/20 0.33
PIM1 P11309 2/20 0.33
SPR P35270 1/20 0.32
LMNA P02545 2/20 0.31
GFER P55789 1/20 0.31
KMT2A Q03164 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CHEK1 O14757 1/20 0.30
CDK2 P24941 1/20 0.30
CSNK2A1 P68400 1/20 0.30
PIM3 Q86V86 1/20 0.30
PIM2 Q9P1W9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20116494 1.00 SLC22A12 (0.35) SLC22A12ADORA2AADORA2BBRAFMAPK3
SCHEMBL20116298 0.75 ADORA2A (0.47) SLC22A12ADORA2AADORA2BBRAFMAPK3
SCHEMBL20660978 0.75 ADORA2A (0.47) SLC22A12ADORA2AADORA2BBRAFMAPK3
SCHEMBL20661130 0.73 SLC22A12 (0.35) SLC22A12ADORA2AADORA2BSPR
SCHEMBL20117306 0.73 ADORA2A (0.47) SLC22A12ADORA2AADORA2BMAPK1SPR
SCHEMBL27259309 0.73 ADORA2A (0.42) SLC22A12ADORA2AADORA2BSPR
SCHEMBL20660789 0.72 ADORA2A (0.47) ADORA2AADORA2BBRAFMAPK3MAPK1
SCHEMBL30506277 0.72 ADORA2A (0.47) ADORA2AADORA2BBRAFMAPK3MAPK1
SCHEMBL20116622 0.72 ADORA2A (0.47) ADORA2AADORA2BBRAFMAPK3MAPK1
SCHEMBL25241798 0.71 LMNA (0.40) LMNAGFERKMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117777121-A Compounds and uses thereof 詹森药业有限公司 2024-03-29 CN disclosed
CN-110099898-B Compounds and uses thereof 优曼尼蒂治疗公司 2023-07-25 CN disclosed