SCHEMBL29045174

SCHEMBL29045174

COc1cc(Cl)nc(OCCCOC(N)=O)c1-c1cc(N)n[nH]1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 3/20 0.47
KCNH2 Q12809 2/20 0.47
HSD17B10 Q99714 2/20 0.36
TNF P01375 1/20 0.33
GAA P10253 1/20 0.33
DYRK1A Q13627 1/20 0.33
CD274 Q9NZQ7 2/20 0.32
PDCD1 Q15116 1/20 0.32
ALDH1A1 P00352 2/20 0.32
LMNA P02545 1/20 0.32
TSHR P16473 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
KDM4E B2RXH2 1/20 0.32
PDCD1LG2 Q9BQ51 1/20 0.31
KMT2A Q03164 2/20 0.31
BCHE P06276 1/20 0.31
ACHE P22303 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29045170 0.83 CHEK1 (0.47) CHEK1KCNH2HSD17B10GAADYRK1A
SCHEMBL24945078 0.82 KCNH2 (0.51) CHEK1KCNH2
SCHEMBL30522689 0.82 KCNH2 (0.51) CHEK1KCNH2
SCHEMBL29045191 0.76 CD274 (0.34) CHEK1KCNH2TNFGAACD274
SCHEMBL29045179 0.71 CHEK1 (0.35) CHEK1KCNH2HSD17B10TNFCD274
SCHEMBL24936161 0.68 KCNH2 (0.66) CHEK1KCNH2DYRK1A
SCHEMBL24485104 0.68 STK17B (0.48) KCNH2
SCHEMBL30522667 0.68 KCNH2 (0.66) CHEK1KCNH2DYRK1A
SCHEMBL24936150 0.64 KCNH2 (0.57) CHEK1KCNH2DYRK1A
SCHEMBL24945515 0.64 KCNH2 (0.49) CHEK1KCNH2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116546974-A 5-heteroaryl-1H-pyrazol-3-amine derivatives 住友制药株式会社 2023-08-04 CN disclosed