SCHEMBL29045191

SCHEMBL29045191

COc1cc(Cl)nc(OCCCOC(N)=O)c1-c1ccno1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 2/20 0.34
PDCD1 Q15116 1/20 0.34
CHEK1 O14757 1/20 0.34
KCNH2 Q12809 1/20 0.34
PDCD1LG2 Q9BQ51 1/20 0.33
TNF P01375 1/20 0.33
BCHE P06276 1/20 0.32
ACHE P22303 1/20 0.32
CYP1A2 P05177 3/20 0.32
CYP19A1 P11511 3/20 0.32
CYP2C9 P11712 3/20 0.32
CYP2C19 P33261 3/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
TSHR P16473 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CYP2D6 P10635 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.31
KMT2A Q03164 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29045194 0.84 CYP1A2 (0.35) CHEK1CYP1A2CYP19A1CYP2C9CYP2C19
SCHEMBL24936246 0.81 KCNH2 (0.43) KCNH2CYP2C19CYP2D6AAK1
SCHEMBL29045174 0.76 CHEK1 (0.47) CD274PDCD1CHEK1KCNH2PDCD1LG2
SCHEMBL29045179 0.71 CHEK1 (0.35) CD274PDCD1CHEK1KCNH2PDCD1LG2
SCHEMBL29827219 0.67 KCNH2 (0.52) KCNH2CYP2C19CYP2D6AAK1
SCHEMBL24936185 0.67 KCNH2 (0.52) KCNH2CYP2C19CYP2D6AAK1
SCHEMBL9818734 0.63 FAAH (0.52) CYP1A2ALDH1A1LMNATSHRL3MBTL1
SCHEMBL29045170 0.62 CHEK1 (0.47) CHEK1KCNH2CYP1A2LMNAKMT2A
SCHEMBL29140637 0.62 MERTK (0.46) LMNAL3MBTL1GAA
SCHEMBL28434588 0.60 CD274 (0.51) CD274PDCD1PDCD1LG2LMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116546974-A 5-heteroaryl-1H-pyrazol-3-amine derivatives 住友制药株式会社 2023-08-04 CN disclosed