SCHEMBL29047862

SCHEMBL29047862

Cc1cc(F)ncc1C(C)O

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.33
CYP2A6 P11509 2/20 0.33
CYP2B6 P20813 2/20 0.33
CYP2C19 P33261 2/20 0.33
APLNR P35414 1/20 0.32
PDE2A O00408 1/20 0.31
FFAR1 O14842 1/20 0.30
AGBL2 Q5U5Z8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24086661 0.86 CYP3A4 (0.33) CYP3A4CYP2A6CYP2B6CYP2C19APLNR
SCHEMBL13315484 0.83 LMNA (0.32) CYP3A4CYP2A6CYP2B6CYP2C19
SCHEMBL23489980 0.79 PDE2A (0.31) PDE2A
SCHEMBL24086587 0.79 PDE2A (0.31) PDE2A
SCHEMBL594120 0.78 PDE2A (0.30) PDE2A
SCHEMBL23489632 0.78 PDE2A (0.44) PDE2A
SCHEMBL16703147 0.76
SCHEMBL23489636 0.76 PDE2A (0.40) PDE2A
SCHEMBL24122426 0.75 ALDH1A1 (0.35) APLNRPDE2A
SCHEMBL13315479 0.72 TLR9 (0.33) CYP3A4CYP2A6CYP2B6CYP2C19FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116157154-A Plasma kallikrein inhibitors 默沙东有限责任公司 2023-05-23 CN disclosed
EP-4178620-A1 PLASMA KALLIKREIN INHIBITORS Merck Sharp & Dohme LLC (US) 2023-05-17 EP disclosed