SCHEMBL29048262

SCHEMBL29048262

O=C(NC1CCN1)c1ccncn1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.53
GRM4 Q14833 3/20 0.44
TNKS O95271 2/20 0.41
GRM5 P41594 1/20 0.38
GSK3A P49840 1/20 0.38
GSK3B P49841 1/20 0.38
RORC P51449 1/20 0.38
ABL1 P00519 1/20 0.38
FAAH O00519 1/20 0.37
CD38 P28907 3/20 0.37
S1PR1 P21453 1/20 0.37
ACKR3 P25106 2/20 0.37
CRBN Q96SW2 1/20 0.36
TNKS2 Q9H2K2 1/20 0.36
CTNNB1 P35222 1/20 0.36
WNT3A P56704 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6645728 0.90 P2RX7 (0.49) P2RX7GRM4TNKSGRM5GSK3A
SCHEMBL9461756 0.89 P2RX7 (0.48) P2RX7GRM4TNKSGRM5GSK3A
SCHEMBL5308759 0.81 P2RX7 (0.51) P2RX7GRM4TNKSGRM5RORC
SCHEMBL7019900 0.77 CD38 (0.57) P2RX7TNKSGRM5CD38S1PR1
SCHEMBL30363652 0.76 P2RX7 (0.53) P2RX7GRM4TNKSGRM5RORC
SCHEMBL25417634 0.75 SMYD3 (0.55) P2RX7TNKSCD38
SCHEMBL29998657 0.75 P2RX7 (0.51) P2RX7GRM4TNKSGRM5RORC
SCHEMBL30336165 0.75 SMYD3 (0.55) P2RX7TNKSCD38
SCHEMBL30338601 0.75 P2RX7 (0.51) P2RX7GRM4TNKSGRM5GSK3A
Hydrochloric Acid SCHEMBL29998785 0.74 P2RX7 (0.50) P2RX7GRM4TNKSGRM5RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116547281-A Isoxazolidines as RIPK1 inhibitors and uses thereof 赛诺菲 2023-08-04 CN disclosed